Assay Detail
Functional
CHEMBL1613763
Review assay metadata, readout intent, target linkage, and publication context from the same page.
PUBCHEM_BIOASSAY: Luminescent dose response cell-based high throughput screening assay for inhibitors of the Janus kinase 2 mutant JAK2V617F. (Class of assay: confirmatory) [Related pubchem assays: 1446 (Primary screen.), 1521 (Confirmation assay.), 1486 (Counter screen.)]
108
Total Activities
108
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Category | confirmatory |
| Confidence | 0 — Uncurated / Unknown |
| Curated By | Autocuration |
Publication
PubChem BioAssay data set
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 108 | 5.92 | 6.65 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL120563 | THIRAM | 2.0 | 1 | 6.65 |
| CHEMBL1973122 | — | — | 1 | 6.65 |
| CHEMBL3191989 | — | — | 1 | 6.63 |
| CHEMBL1572967 | — | — | 1 | 6.46 |
| CHEMBL1427185 | — | — | 1 | 6.42 |
| CHEMBL1543839 | — | — | 1 | 6.40 |
| CHEMBL3193058 | — | — | 1 | 6.36 |
| CHEMBL1424118 | — | — | 1 | 6.32 |
| CHEMBL1520801 | — | — | 1 | 6.27 |
| CHEMBL1450393 | — | — | 1 | 6.25 |
| CHEMBL1304902 | — | — | 1 | 6.24 |
| CHEMBL1423501 | — | — | 1 | 6.22 |
| CHEMBL1466500 | — | — | 1 | 6.22 |
| CHEMBL1341981 | — | — | 1 | 6.20 |
| CHEMBL1318943 | — | — | 1 | 6.20 |
| CHEMBL1447125 | — | — | 1 | 6.20 |
| CHEMBL1399938 | — | — | 1 | 6.19 |
| CHEMBL1444859 | — | — | 1 | 6.19 |
| CHEMBL1470728 | — | — | 1 | 6.19 |
| CHEMBL1299997 | — | — | 1 | 6.18 |
| CHEMBL1459746 | — | — | 1 | 6.17 |
| CHEMBL1613090 | — | — | 1 | 6.17 |
| CHEMBL1449794 | — | — | 1 | 6.16 |
| CHEMBL1440303 | — | — | 1 | 6.15 |
| CHEMBL1524240 | — | — | 1 | 6.15 |
| CHEMBL1481030 | — | — | 1 | 6.14 |
| CHEMBL1585185 | — | — | 1 | 6.14 |
| CHEMBL1597039 | — | — | 1 | 6.13 |
| CHEMBL1980982 | — | — | 1 | 6.13 |
| CHEMBL1482285 | — | — | 1 | 6.12 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL120563 | THIRAM | IC50 | = | 223.0 | nM | 6.65 |
| CHEMBL1973122 | — | IC50 | = | 224.0 | nM | 6.65 |
| CHEMBL3191989 | — | IC50 | = | 235.0 | nM | 6.63 |
| CHEMBL1572967 | — | IC50 | = | 351.0 | nM | 6.46 |
| CHEMBL1427185 | — | IC50 | = | 383.0 | nM | 6.42 |
| CHEMBL1543839 | — | IC50 | = | 401.0 | nM | 6.40 |
| CHEMBL3193058 | — | IC50 | = | 442.0 | nM | 6.36 |
| CHEMBL1424118 | — | IC50 | = | 476.0 | nM | 6.32 |
| CHEMBL1520801 | — | IC50 | = | 542.0 | nM | 6.27 |
| CHEMBL1450393 | — | IC50 | = | 562.0 | nM | 6.25 |
| CHEMBL1304902 | — | IC50 | = | 581.0 | nM | 6.24 |
| CHEMBL1466500 | — | IC50 | = | 597.0 | nM | 6.22 |
| CHEMBL1423501 | — | IC50 | = | 605.0 | nM | 6.22 |
| CHEMBL1447125 | — | IC50 | = | 628.0 | nM | 6.20 |
| CHEMBL1341981 | — | IC50 | = | 632.0 | nM | 6.20 |
| CHEMBL1318943 | — | IC50 | = | 637.0 | nM | 6.20 |
| CHEMBL1470728 | — | IC50 | = | 639.0 | nM | 6.19 |
| CHEMBL1399938 | — | IC50 | = | 649.0 | nM | 6.19 |
| CHEMBL1444859 | — | IC50 | = | 644.0 | nM | 6.19 |
| CHEMBL1299997 | — | IC50 | = | 653.0 | nM | 6.18 |
| CHEMBL1613090 | — | IC50 | = | 676.0 | nM | 6.17 |
| CHEMBL1459746 | — | IC50 | = | 670.0 | nM | 6.17 |
| CHEMBL1449794 | — | IC50 | = | 695.0 | nM | 6.16 |
| CHEMBL1524240 | — | IC50 | = | 702.0 | nM | 6.15 |
| CHEMBL1440303 | — | IC50 | = | 707.0 | nM | 6.15 |
| CHEMBL1585185 | — | IC50 | = | 730.0 | nM | 6.14 |
| CHEMBL1481030 | — | IC50 | = | 721.0 | nM | 6.14 |
| CHEMBL1597039 | — | IC50 | = | 743.0 | nM | 6.13 |
| CHEMBL1980982 | — | IC50 | = | 744.0 | nM | 6.13 |
| CHEMBL1482285 | — | IC50 | = | 768.0 | nM | 6.12 |
| CHEMBL1549175 | — | IC50 | = | 788.0 | nM | 6.10 |
| CHEMBL1557820 | — | IC50 | = | 787.0 | nM | 6.10 |
| CHEMBL1439384 | — | IC50 | = | 810.0 | nM | 6.09 |
| CHEMBL585 | TRIAMTERENE | IC50 | = | 807.0 | nM | 6.09 |
| CHEMBL1511663 | — | IC50 | = | 835.0 | nM | 6.08 |
| CHEMBL1365696 | — | IC50 | = | 826.0 | nM | 6.08 |
| CHEMBL1427637 | — | IC50 | = | 824.0 | nM | 6.08 |
| CHEMBL1305275 | — | IC50 | = | 870.0 | nM | 6.06 |
| CHEMBL1470321 | — | IC50 | = | 870.0 | nM | 6.06 |
| CHEMBL1382022 | — | IC50 | = | 909.0 | nM | 6.04 |
| CHEMBL1476181 | — | IC50 | = | 934.0 | nM | 6.03 |
| CHEMBL1562235 | — | IC50 | = | 960.0 | nM | 6.02 |
| CHEMBL1574219 | — | IC50 | = | 996.0 | nM | 6.00 |
| CHEMBL1393319 | — | IC50 | = | 1030.0 | nM | 5.99 |
| CHEMBL1498517 | — | IC50 | = | 1025.0 | nM | 5.99 |
| CHEMBL1478382 | — | IC50 | = | 1023.0 | nM | 5.99 |
| CHEMBL1466593 | — | IC50 | = | 1058.0 | nM | 5.98 |
| CHEMBL1597766 | — | IC50 | = | 1102.0 | nM | 5.96 |
| CHEMBL1981883 | — | IC50 | = | 1149.0 | nM | 5.94 |
| CHEMBL1411125 | — | IC50 | = | 1148.0 | nM | 5.94 |