Assay Detail
Binding
CHEMBL1613774
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PUBCHEM_BIOASSAY: Confirmation of compounds inhibiting phosphomannose isomerase (PMI) via a fluorescence intensity assay using a high concentration of mannose 6-phosphate. (Class of assay: confirmatory) [Related pubchem assays (depositor defined):AID1209, AID1220, AID1545, AID1553, AID1620]
16
Total Activities
13
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Category | confirmatory |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
PubChem BioAssay data set
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 16 | 4.90 | 5.26 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL1449845 | — | — | 1 | 5.26 |
| CHEMBL1369613 | — | — | 1 | 4.85 |
| CHEMBL1339149 | — | — | 1 | 4.79 |
| CHEMBL45152 | — | — | 1 | 4.68 |
| CHEMBL1479664 | — | — | 1 | - |
| CHEMBL1333813 | — | — | 2 | - |
| CHEMBL1569077 | — | — | 1 | - |
| CHEMBL1443661 | — | — | 1 | - |
| CHEMBL1606954 | — | — | 1 | - |
| CHEMBL1300370 | — | — | 2 | - |
| CHEMBL1520471 | — | — | 2 | - |
| CHEMBL1531603 | — | — | 1 | - |
| CHEMBL1609086 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL1449845 | — | IC50 | = | 5510.0 | nM | 5.26 |
| CHEMBL1369613 | — | IC50 | = | 14000.0 | nM | 4.85 |
| CHEMBL1339149 | — | IC50 | = | 16400.0 | nM | 4.79 |
| CHEMBL45152 | — | IC50 | = | 21000.0 | nM | 4.68 |
| CHEMBL1479664 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL1333813 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL1569077 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL1443661 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL1333813 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL1606954 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL1300370 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL1520471 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL1520471 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL1300370 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL1531603 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL1609086 | — | IC50 | > | 100000.0 | nM | - |