Assay Detail
Functional
CHEMBL1613794
Review assay metadata, readout intent, target linkage, and publication context from the same page.
PUBCHEM_BIOASSAY: Fluorescence Cell-Based Secondary Assay for toxicity in mammalian fibroblasts. (Class of assay: confirmatory) [Related pubchem assays (depositor defined):AID1979, AID2007]
1833
Total Activities
1830
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Category | confirmatory |
| Confidence | 0 — Uncurated / Unknown |
| Curated By | Autocuration |
Publication
PubChem BioAssay data set
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| EC50 | 1833 | 4.75 | 6.75 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL1200976 | IDARUBICIN HYDROCHLORIDE | 4.0 | 1 | 6.75 |
| CHEMBL300389 | — | — | 1 | 6.57 |
| CHEMBL599924 | — | — | 1 | 6.02 |
| CHEMBL1985582 | — | — | 1 | 6.00 |
| CHEMBL1383334 | — | — | 1 | 5.92 |
| CHEMBL89445 | TERPYRIDINE | — | 1 | 5.88 |
| CHEMBL1392643 | — | — | 1 | 5.83 |
| CHEMBL1543257 | — | — | 1 | 5.80 |
| CHEMBL3199020 | — | — | 1 | 5.79 |
| CHEMBL1452795 | — | — | 1 | 5.77 |
| CHEMBL586135 | — | — | 1 | 5.75 |
| CHEMBL1488035 | — | — | 1 | 5.74 |
| CHEMBL1572967 | — | — | 1 | 5.73 |
| CHEMBL1544131 | — | — | 1 | 5.64 |
| CHEMBL3145303 | — | — | 1 | 5.63 |
| CHEMBL3192995 | — | — | 1 | 5.62 |
| CHEMBL1470149 | — | — | 1 | 5.62 |
| CHEMBL3198720 | — | — | 1 | 5.60 |
| CHEMBL1543839 | — | — | 1 | 5.59 |
| CHEMBL1543977 | — | — | 1 | 5.59 |
| CHEMBL1387177 | — | — | 1 | 5.59 |
| CHEMBL1606097 | — | — | 1 | 5.59 |
| CHEMBL3199737 | — | — | 1 | 5.59 |
| CHEMBL1519576 | — | — | 1 | 5.59 |
| CHEMBL3191763 | — | — | 1 | 5.59 |
| CHEMBL1337500 | — | — | 1 | 5.58 |
| CHEMBL1341270 | — | — | 1 | 5.58 |
| CHEMBL2095095 | — | — | 1 | 5.58 |
| CHEMBL1451931 | — | — | 1 | 5.58 |
| CHEMBL3198723 | — | — | 1 | 5.57 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL1200976 | IDARUBICIN HYDROCHLORIDE | EC50 | = | 178.0 | nM | 6.75 |
| CHEMBL300389 | — | EC50 | = | 269.0 | nM | 6.57 |
| CHEMBL599924 | — | EC50 | = | 952.0 | nM | 6.02 |
| CHEMBL1985582 | — | EC50 | = | 1009.0 | nM | 6.00 |
| CHEMBL1383334 | — | EC50 | = | 1211.0 | nM | 5.92 |
| CHEMBL89445 | TERPYRIDINE | EC50 | = | 1324.0 | nM | 5.88 |
| CHEMBL1392643 | — | EC50 | = | 1479.0 | nM | 5.83 |
| CHEMBL1543257 | — | EC50 | = | 1600.0 | nM | 5.80 |
| CHEMBL3199020 | — | EC50 | = | 1608.0 | nM | 5.79 |
| CHEMBL1452795 | — | EC50 | = | 1707.0 | nM | 5.77 |
| CHEMBL586135 | — | EC50 | = | 1762.0 | nM | 5.75 |
| CHEMBL1488035 | — | EC50 | = | 1801.0 | nM | 5.74 |
| CHEMBL1572967 | — | EC50 | = | 1846.0 | nM | 5.73 |
| CHEMBL1544131 | — | EC50 | = | 2268.0 | nM | 5.64 |
| CHEMBL3145303 | — | EC50 | = | 2318.0 | nM | 5.63 |
| CHEMBL1470149 | — | EC50 | = | 2376.0 | nM | 5.62 |
| CHEMBL3192995 | — | EC50 | = | 2373.0 | nM | 5.62 |
| CHEMBL3198720 | — | EC50 | = | 2495.0 | nM | 5.60 |
| CHEMBL1543839 | — | EC50 | = | 2568.0 | nM | 5.59 |
| CHEMBL1387177 | — | EC50 | = | 2558.0 | nM | 5.59 |
| CHEMBL3199737 | — | EC50 | = | 2548.0 | nM | 5.59 |
| CHEMBL1543977 | — | EC50 | = | 2590.0 | nM | 5.59 |
| CHEMBL1606097 | — | EC50 | = | 2541.0 | nM | 5.59 |
| CHEMBL1519576 | — | EC50 | = | 2592.0 | nM | 5.59 |
| CHEMBL3191763 | — | EC50 | = | 2547.0 | nM | 5.59 |
| CHEMBL2095095 | — | EC50 | = | 2657.0 | nM | 5.58 |
| CHEMBL1341270 | — | EC50 | = | 2613.0 | nM | 5.58 |
| CHEMBL1337500 | — | EC50 | = | 2656.0 | nM | 5.58 |
| CHEMBL1451931 | — | EC50 | = | 2610.0 | nM | 5.58 |
| CHEMBL3198723 | — | EC50 | = | 2668.0 | nM | 5.57 |
| CHEMBL3190594 | — | EC50 | = | 2705.0 | nM | 5.57 |
| CHEMBL1449040 | — | EC50 | = | 2674.0 | nM | 5.57 |
| CHEMBL1605956 | — | EC50 | = | 2690.0 | nM | 5.57 |
| CHEMBL1563714 | — | EC50 | = | 2667.0 | nM | 5.57 |
| CHEMBL199868 | — | EC50 | = | 2763.0 | nM | 5.56 |
| CHEMBL3197076 | — | EC50 | = | 2858.0 | nM | 5.54 |
| CHEMBL1441218 | — | EC50 | = | 2972.0 | nM | 5.53 |
| CHEMBL1536643 | — | EC50 | = | 2934.0 | nM | 5.53 |
| CHEMBL1569910 | — | EC50 | = | 3010.0 | nM | 5.52 |
| CHEMBL1380406 | — | EC50 | = | 3042.0 | nM | 5.52 |
| CHEMBL1343392 | — | EC50 | = | 3069.0 | nM | 5.51 |
| CHEMBL1887153 | — | EC50 | = | 3173.0 | nM | 5.50 |
| CHEMBL601543 | — | EC50 | = | 3159.0 | nM | 5.50 |
| CHEMBL3197978 | — | EC50 | = | 3134.0 | nM | 5.50 |
| CHEMBL1463847 | — | EC50 | = | 3150.0 | nM | 5.50 |
| CHEMBL469036 | ENNIATIN B | EC50 | = | 3219.0 | nM | 5.49 |
| CHEMBL1377849 | — | EC50 | = | 3252.0 | nM | 5.49 |
| CHEMBL1993194 | — | EC50 | = | 3291.0 | nM | 5.48 |
| CHEMBL1440300 | — | EC50 | = | 3496.0 | nM | 5.46 |
| CHEMBL1370513 | — | EC50 | = | 3586.0 | nM | 5.45 |