Assay Detail
Functional
CHEMBL1613987
Review assay metadata, readout intent, target linkage, and publication context from the same page.
PUBCHEM_BIOASSAY: Luminescence Cell-Based Dose HTS Response to Identify Inhibitors of 5'UTR Stem-Loop Driven Prion Protein mRNA Translation in H4-C Neuroglioblastoma Cells. (Class of assay: confirmatory) [Related pubchem assays (depositor defined):AID1814, AID1827]
28
Total Activities
28
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Category | confirmatory |
| Confidence | 0 — Uncurated / Unknown |
| Curated By | Autocuration |
Publication
PubChem BioAssay data set
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| EC50 | 28 | 5.92 | 6.79 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL1331904 | — | — | 1 | 6.79 |
| CHEMBL1371056 | — | — | 1 | 6.73 |
| CHEMBL1331733 | — | — | 1 | 6.62 |
| CHEMBL1493731 | — | — | 1 | 6.49 |
| CHEMBL1389580 | — | — | 1 | 6.33 |
| CHEMBL1349455 | — | — | 1 | 6.23 |
| CHEMBL1522289 | — | — | 1 | 6.16 |
| CHEMBL1354131 | — | — | 1 | 6.15 |
| CHEMBL1313968 | — | — | 1 | 6.14 |
| CHEMBL1476264 | — | — | 1 | 6.04 |
| CHEMBL1316021 | — | — | 1 | 5.96 |
| CHEMBL1330793 | — | — | 1 | 5.95 |
| CHEMBL1528120 | — | — | 1 | 5.94 |
| CHEMBL1513325 | — | — | 1 | 5.91 |
| CHEMBL1314043 | — | — | 1 | 5.81 |
| CHEMBL1569667 | — | — | 1 | 5.77 |
| CHEMBL1358278 | — | — | 1 | 5.76 |
| CHEMBL1354093 | — | — | 1 | 5.75 |
| CHEMBL602722 | — | — | 1 | 5.71 |
| CHEMBL1408486 | — | — | 1 | 5.63 |
| CHEMBL1331836 | — | — | 1 | 5.62 |
| CHEMBL1555236 | — | — | 1 | 5.62 |
| CHEMBL1620207 | — | — | 1 | 5.53 |
| CHEMBL1440659 | — | — | 1 | 5.45 |
| CHEMBL1407944 | — | — | 1 | 5.23 |
| CHEMBL1300558 | — | — | 1 | 4.65 |
| CHEMBL1490480 | — | — | 1 | - |
| CHEMBL1412667 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL1331904 | — | EC50 | = | 162.0 | nM | 6.79 |
| CHEMBL1371056 | — | EC50 | = | 186.0 | nM | 6.73 |
| CHEMBL1331733 | — | EC50 | = | 241.0 | nM | 6.62 |
| CHEMBL1493731 | — | EC50 | = | 325.0 | nM | 6.49 |
| CHEMBL1389580 | — | EC50 | = | 464.0 | nM | 6.33 |
| CHEMBL1349455 | — | EC50 | = | 592.0 | nM | 6.23 |
| CHEMBL1522289 | — | EC50 | = | 699.0 | nM | 6.16 |
| CHEMBL1354131 | — | EC50 | = | 711.0 | nM | 6.15 |
| CHEMBL1313968 | — | EC50 | = | 722.0 | nM | 6.14 |
| CHEMBL1476264 | — | EC50 | = | 904.0 | nM | 6.04 |
| CHEMBL1316021 | — | EC50 | = | 1090.0 | nM | 5.96 |
| CHEMBL1330793 | — | EC50 | = | 1129.0 | nM | 5.95 |
| CHEMBL1528120 | — | EC50 | = | 1147.0 | nM | 5.94 |
| CHEMBL1513325 | — | EC50 | = | 1232.0 | nM | 5.91 |
| CHEMBL1314043 | — | EC50 | = | 1541.0 | nM | 5.81 |
| CHEMBL1569667 | — | EC50 | = | 1686.0 | nM | 5.77 |
| CHEMBL1358278 | — | EC50 | = | 1754.0 | nM | 5.76 |
| CHEMBL1354093 | — | EC50 | = | 1760.0 | nM | 5.75 |
| CHEMBL602722 | — | EC50 | = | 1948.0 | nM | 5.71 |
| CHEMBL1408486 | — | EC50 | = | 2326.0 | nM | 5.63 |
| CHEMBL1331836 | — | EC50 | = | 2399.0 | nM | 5.62 |
| CHEMBL1555236 | — | EC50 | = | 2399.0 | nM | 5.62 |
| CHEMBL1620207 | — | EC50 | = | 2937.0 | nM | 5.53 |
| CHEMBL1440659 | — | EC50 | = | 3561.0 | nM | 5.45 |
| CHEMBL1407944 | — | EC50 | = | 5897.0 | nM | 5.23 |
| CHEMBL1300558 | — | EC50 | = | 22448.0 | nM | 4.65 |
| CHEMBL1490480 | — | EC50 | > | 195000.0 | nM | - |
| CHEMBL1412667 | — | EC50 | > | 195000.0 | nM | - |