Assay Detail
Functional
CHEMBL1613998
Review assay metadata, readout intent, target linkage, and publication context from the same page.
PUBCHEM_BIOASSAY: Luminescent counterscreen for inhibitors of the Janus kinase 2 mutant JAK2V617F: dose response cell-based high throughput screening assay for inhibitors of parental Ba/F3 cell viability. (Class of assay: confirmatory) [Related pubchem assays: 1446 (Primary screen.), 1486 (Counterscreen in triplicate.), 1691 (Dose response.)]
108
Total Activities
108
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Cell Type | BaF3 |
| Category | confirmatory |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
PubChem BioAssay data set
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 108 | 5.37 | 6.65 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL120563 | THIRAM | 2.0 | 1 | 6.65 |
| CHEMBL3191989 | — | — | 1 | 6.18 |
| CHEMBL1973122 | — | — | 1 | 5.99 |
| CHEMBL1424118 | — | — | 1 | 5.97 |
| CHEMBL3193058 | — | — | 1 | 5.96 |
| CHEMBL1572967 | — | — | 1 | 5.94 |
| CHEMBL1543839 | — | — | 1 | 5.92 |
| CHEMBL1481030 | — | — | 1 | 5.90 |
| CHEMBL1304902 | — | — | 1 | 5.87 |
| CHEMBL1364913 | — | — | 1 | 5.85 |
| CHEMBL1459746 | — | — | 1 | 5.82 |
| CHEMBL1399938 | — | — | 1 | 5.79 |
| CHEMBL1341981 | — | — | 1 | 5.78 |
| CHEMBL3193428 | — | — | 1 | 5.78 |
| CHEMBL1427637 | — | — | 1 | 5.77 |
| CHEMBL1427185 | — | — | 1 | 5.75 |
| CHEMBL1466500 | — | — | 1 | 5.72 |
| CHEMBL1447125 | — | — | 1 | 5.68 |
| CHEMBL1482285 | — | — | 1 | 5.68 |
| CHEMBL1379604 | — | — | 1 | 5.67 |
| CHEMBL1440303 | — | — | 1 | 5.65 |
| CHEMBL1444859 | — | — | 1 | 5.64 |
| CHEMBL1585185 | — | — | 1 | 5.62 |
| CHEMBL1382022 | — | — | 1 | 5.61 |
| CHEMBL1423501 | — | — | 1 | 5.60 |
| CHEMBL1521348 | — | — | 1 | 5.58 |
| CHEMBL1597766 | — | — | 1 | 5.55 |
| CHEMBL1557820 | — | — | 1 | 5.54 |
| CHEMBL1560296 | — | — | 1 | 5.53 |
| CHEMBL1518085 | — | — | 1 | 5.52 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL120563 | THIRAM | IC50 | = | 223.0 | nM | 6.65 |
| CHEMBL3191989 | — | IC50 | = | 653.0 | nM | 6.18 |
| CHEMBL1973122 | — | IC50 | = | 1036.0 | nM | 5.99 |
| CHEMBL1424118 | — | IC50 | = | 1081.0 | nM | 5.97 |
| CHEMBL3193058 | — | IC50 | = | 1110.0 | nM | 5.96 |
| CHEMBL1572967 | — | IC50 | = | 1138.0 | nM | 5.94 |
| CHEMBL1543839 | — | IC50 | = | 1199.0 | nM | 5.92 |
| CHEMBL1481030 | — | IC50 | = | 1263.0 | nM | 5.90 |
| CHEMBL1304902 | — | IC50 | = | 1342.0 | nM | 5.87 |
| CHEMBL1364913 | — | IC50 | = | 1421.0 | nM | 5.85 |
| CHEMBL1459746 | — | IC50 | = | 1500.0 | nM | 5.82 |
| CHEMBL1399938 | — | IC50 | = | 1631.0 | nM | 5.79 |
| CHEMBL1341981 | — | IC50 | = | 1676.0 | nM | 5.78 |
| CHEMBL3193428 | — | IC50 | = | 1666.0 | nM | 5.78 |
| CHEMBL1427637 | — | IC50 | = | 1711.0 | nM | 5.77 |
| CHEMBL1427185 | — | IC50 | = | 1760.0 | nM | 5.75 |
| CHEMBL1466500 | — | IC50 | = | 1924.0 | nM | 5.72 |
| CHEMBL1447125 | — | IC50 | = | 2072.0 | nM | 5.68 |
| CHEMBL1482285 | — | IC50 | = | 2067.0 | nM | 5.68 |
| CHEMBL1379604 | — | IC50 | = | 2113.0 | nM | 5.67 |
| CHEMBL1440303 | — | IC50 | = | 2259.0 | nM | 5.65 |
| CHEMBL1444859 | — | IC50 | = | 2283.0 | nM | 5.64 |
| CHEMBL1585185 | — | IC50 | = | 2404.0 | nM | 5.62 |
| CHEMBL1382022 | — | IC50 | = | 2460.0 | nM | 5.61 |
| CHEMBL1423501 | — | IC50 | = | 2506.0 | nM | 5.60 |
| CHEMBL1521348 | — | IC50 | = | 2656.0 | nM | 5.58 |
| CHEMBL1597766 | — | IC50 | = | 2833.0 | nM | 5.55 |
| CHEMBL1557820 | — | IC50 | = | 2906.0 | nM | 5.54 |
| CHEMBL1560296 | — | IC50 | = | 2966.0 | nM | 5.53 |
| CHEMBL1518085 | — | IC50 | = | 3020.0 | nM | 5.52 |
| CHEMBL1563340 | — | IC50 | = | 3125.0 | nM | 5.50 |
| CHEMBL1439384 | — | IC50 | = | 3261.0 | nM | 5.49 |
| CHEMBL254255 | — | IC50 | = | 3336.0 | nM | 5.48 |
| CHEMBL1489454 | — | IC50 | = | 3341.0 | nM | 5.48 |
| CHEMBL1501466 | — | IC50 | = | 3311.0 | nM | 5.48 |
| CHEMBL1299997 | — | IC50 | = | 3498.0 | nM | 5.46 |
| CHEMBL1476181 | — | IC50 | = | 3503.0 | nM | 5.46 |
| CHEMBL1334315 | — | IC50 | = | 3565.0 | nM | 5.45 |
| CHEMBL3214200 | — | IC50 | = | 3619.0 | nM | 5.44 |
| CHEMBL1470321 | — | IC50 | = | 3644.0 | nM | 5.44 |
| CHEMBL1411125 | — | IC50 | = | 3615.0 | nM | 5.44 |
| CHEMBL1431684 | — | IC50 | = | 3676.0 | nM | 5.43 |
| CHEMBL1549175 | — | IC50 | = | 3741.0 | nM | 5.43 |
| CHEMBL1599994 | — | IC50 | = | 3699.0 | nM | 5.43 |
| CHEMBL1525669 | — | IC50 | = | 3759.0 | nM | 5.42 |
| CHEMBL1470728 | — | IC50 | = | 3850.0 | nM | 5.42 |
| CHEMBL1466593 | — | IC50 | = | 4217.0 | nM | 5.38 |
| CHEMBL1393319 | — | IC50 | = | 4277.0 | nM | 5.37 |
| CHEMBL1305275 | — | IC50 | = | 4373.0 | nM | 5.36 |
| CHEMBL1562235 | — | IC50 | = | 4387.0 | nM | 5.36 |