Assay Detail
Functional
CHEMBL1614025
Review assay metadata, readout intent, target linkage, and publication context from the same page.
PUBCHEM_BIOASSAY: Late stage counterscreen assay for S1P4 antagonists: Fluorescence dose response cell-based screening assay for antagonists of the Sphingosine 1-Phosphate Receptor 1 (S1P1). (Class of assay: confirmatory) [Related pubchem assays (depositor defined):AID1510, AID1524, AID1692, AID1853, AID2332, AID489009, AID489017]
21
Total Activities
21
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Category | confirmatory |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
PubChem BioAssay data set
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 21 | 5.75 | 6.46 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL1412583 | — | — | 1 | 6.46 |
| CHEMBL1592119 | — | — | 1 | 5.03 |
| CHEMBL1472539 | — | — | 1 | - |
| CHEMBL1393993 | — | — | 1 | - |
| CHEMBL1589684 | — | — | 1 | - |
| CHEMBL1514981 | — | — | 1 | - |
| CHEMBL1603615 | — | — | 1 | - |
| CHEMBL1393906 | — | — | 1 | - |
| CHEMBL1316334 | — | — | 1 | - |
| CHEMBL1592813 | — | — | 1 | - |
| CHEMBL1415555 | — | — | 1 | - |
| CHEMBL1354080 | — | — | 1 | - |
| CHEMBL1397874 | — | — | 1 | - |
| CHEMBL1354895 | — | — | 1 | - |
| CHEMBL1436066 | — | — | 1 | - |
| CHEMBL1331049 | — | — | 1 | - |
| CHEMBL1511831 | — | — | 1 | - |
| CHEMBL1511839 | — | — | 1 | - |
| CHEMBL1553396 | — | — | 1 | - |
| CHEMBL1473443 | — | — | 1 | - |
| CHEMBL1550998 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL1412583 | — | IC50 | = | 351.0 | nM | 6.46 |
| CHEMBL1592119 | — | IC50 | = | 9312.0 | nM | 5.03 |
| CHEMBL1472539 | — | IC50 | > | 25000.0 | nM | - |
| CHEMBL1393993 | — | IC50 | > | 25000.0 | nM | - |
| CHEMBL1589684 | — | IC50 | > | 25000.0 | nM | - |
| CHEMBL1514981 | — | IC50 | > | 25000.0 | nM | - |
| CHEMBL1603615 | — | IC50 | > | 25000.0 | nM | - |
| CHEMBL1393906 | — | IC50 | > | 25000.0 | nM | - |
| CHEMBL1316334 | — | IC50 | > | 25000.0 | nM | - |
| CHEMBL1592813 | — | IC50 | > | 25000.0 | nM | - |
| CHEMBL1415555 | — | IC50 | > | 25000.0 | nM | - |
| CHEMBL1354080 | — | IC50 | > | 25000.0 | nM | - |
| CHEMBL1397874 | — | IC50 | > | 25000.0 | nM | - |
| CHEMBL1354895 | — | IC50 | > | 25000.0 | nM | - |
| CHEMBL1436066 | — | IC50 | > | 25000.0 | nM | - |
| CHEMBL1331049 | — | IC50 | > | 25000.0 | nM | - |
| CHEMBL1511831 | — | IC50 | > | 25000.0 | nM | - |
| CHEMBL1511839 | — | IC50 | > | 25000.0 | nM | - |
| CHEMBL1553396 | — | IC50 | > | 25000.0 | nM | - |
| CHEMBL1473443 | — | IC50 | > | 25000.0 | nM | - |
| CHEMBL1550998 | — | IC50 | > | 25000.0 | nM | - |