Assay Detail
Functional
CHEMBL1614083
Review assay metadata, readout intent, target linkage, and publication context from the same page.
PUBCHEM_BIOASSAY: Fluorescence-based counterscreen for antagonists of the G-protein coupled receptor 7 (GPR7): cell-based high throughput dose response assay to identify antagonists of the melanin-concentrating hormone receptor 1 (MCHR1). (Class of assay: confirmatory) [Related pubchem assays: 1880 (Summary AID.), 2148 (Screening assay (MCHR1 antagonists).), 1952 (Screening assay (GPR7 antagonists).), 1861 (Screening assay (GPR7 antagonists).)]
126
Total Activities
126
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Category | confirmatory |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Target
Melanin-concentrating hormone receptor 1 (CHEMBL344) ↗| Type | SINGLE PROTEIN |
| Organism | Homo sapiens |
Publication
PubChem BioAssay data set
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 126 | 4.75 | 5.32 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL1484343 | — | — | 1 | 5.32 |
| CHEMBL1582334 | — | — | 1 | 5.18 |
| CHEMBL1458112 | — | — | 1 | 5.10 |
| CHEMBL1549996 | — | — | 1 | 5.07 |
| CHEMBL1568072 | — | — | 1 | 5.03 |
| CHEMBL1401638 | — | — | 1 | 5.00 |
| CHEMBL1412874 | — | — | 1 | 4.98 |
| CHEMBL1436519 | — | — | 1 | 4.97 |
| CHEMBL1319565 | — | — | 1 | 4.95 |
| CHEMBL1332346 | — | — | 1 | 4.95 |
| CHEMBL1589201 | — | — | 1 | 4.95 |
| CHEMBL1359426 | — | — | 1 | 4.92 |
| CHEMBL1499675 | — | — | 1 | 4.92 |
| CHEMBL1585038 | — | — | 1 | 4.92 |
| CHEMBL1342885 | — | — | 1 | 4.90 |
| CHEMBL1533829 | — | — | 1 | 4.90 |
| CHEMBL1576145 | — | — | 1 | 4.90 |
| CHEMBL1339438 | — | — | 1 | 4.89 |
| CHEMBL1977747 | — | — | 1 | 4.89 |
| CHEMBL1537947 | — | — | 1 | 4.88 |
| CHEMBL1471999 | — | — | 1 | 4.88 |
| CHEMBL1335685 | — | — | 1 | 4.83 |
| CHEMBL1609915 | — | — | 1 | 4.82 |
| CHEMBL1467280 | — | — | 1 | 4.82 |
| CHEMBL1359489 | — | — | 1 | 4.80 |
| CHEMBL1595687 | — | — | 1 | 4.80 |
| CHEMBL1578660 | — | — | 1 | 4.80 |
| CHEMBL1569862 | — | — | 1 | 4.80 |
| CHEMBL1582511 | — | — | 1 | 4.80 |
| CHEMBL1350024 | — | — | 1 | 4.79 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL1484343 | — | IC50 | = | 4756.0 | nM | 5.32 |
| CHEMBL1582334 | — | IC50 | = | 6596.0 | nM | 5.18 |
| CHEMBL1458112 | — | IC50 | = | 8010.0 | nM | 5.10 |
| CHEMBL1549996 | — | IC50 | = | 8434.0 | nM | 5.07 |
| CHEMBL1568072 | — | IC50 | = | 9305.0 | nM | 5.03 |
| CHEMBL1401638 | — | IC50 | = | 9960.0 | nM | 5.00 |
| CHEMBL1412874 | — | IC50 | = | 10409.0 | nM | 4.98 |
| CHEMBL1436519 | — | IC50 | = | 10598.0 | nM | 4.97 |
| CHEMBL1589201 | — | IC50 | = | 11254.0 | nM | 4.95 |
| CHEMBL1319565 | — | IC50 | = | 11162.0 | nM | 4.95 |
| CHEMBL1332346 | — | IC50 | = | 11115.0 | nM | 4.95 |
| CHEMBL1499675 | — | IC50 | = | 11900.0 | nM | 4.92 |
| CHEMBL1585038 | — | IC50 | = | 12134.0 | nM | 4.92 |
| CHEMBL1359426 | — | IC50 | = | 12007.0 | nM | 4.92 |
| CHEMBL1576145 | — | IC50 | = | 12631.0 | nM | 4.90 |
| CHEMBL1533829 | — | IC50 | = | 12520.0 | nM | 4.90 |
| CHEMBL1342885 | — | IC50 | = | 12573.0 | nM | 4.90 |
| CHEMBL1339438 | — | IC50 | = | 12956.0 | nM | 4.89 |
| CHEMBL1977747 | — | IC50 | = | 13012.0 | nM | 4.89 |
| CHEMBL1471999 | — | IC50 | = | 13298.0 | nM | 4.88 |
| CHEMBL1537947 | — | IC50 | = | 13334.0 | nM | 4.88 |
| CHEMBL1335685 | — | IC50 | = | 14706.0 | nM | 4.83 |
| CHEMBL1467280 | — | IC50 | = | 15017.0 | nM | 4.82 |
| CHEMBL1609915 | — | IC50 | = | 15007.0 | nM | 4.82 |
| CHEMBL1595687 | — | IC50 | = | 16012.0 | nM | 4.80 |
| CHEMBL1569862 | — | IC50 | = | 15852.0 | nM | 4.80 |
| CHEMBL1578660 | — | IC50 | = | 15693.0 | nM | 4.80 |
| CHEMBL1359489 | — | IC50 | = | 15954.0 | nM | 4.80 |
| CHEMBL1582511 | — | IC50 | = | 15875.0 | nM | 4.80 |
| CHEMBL1350024 | — | IC50 | = | 16167.0 | nM | 4.79 |
| CHEMBL1586617 | — | IC50 | = | 16568.0 | nM | 4.78 |
| CHEMBL1343746 | — | IC50 | = | 16555.0 | nM | 4.78 |
| CHEMBL1418691 | — | IC50 | = | 16860.0 | nM | 4.77 |
| CHEMBL1539046 | — | IC50 | = | 17127.0 | nM | 4.77 |
| CHEMBL1314041 | — | IC50 | = | 17646.0 | nM | 4.75 |
| CHEMBL1538063 | — | IC50 | = | 18266.0 | nM | 4.74 |
| CHEMBL1480448 | — | IC50 | = | 18854.0 | nM | 4.72 |
| CHEMBL1312413 | — | IC50 | = | 19561.0 | nM | 4.71 |
| CHEMBL1573548 | — | IC50 | = | 20045.0 | nM | 4.70 |
| CHEMBL1461182 | — | IC50 | = | 19848.0 | nM | 4.70 |
| CHEMBL1446321 | — | IC50 | = | 20714.0 | nM | 4.68 |
| CHEMBL1353612 | — | IC50 | = | 21512.0 | nM | 4.67 |
| CHEMBL1358809 | — | IC50 | = | 21793.0 | nM | 4.66 |
| CHEMBL1493564 | — | IC50 | = | 22190.0 | nM | 4.65 |
| CHEMBL1518183 | — | IC50 | = | 22792.0 | nM | 4.64 |
| CHEMBL1447678 | — | IC50 | = | 22951.0 | nM | 4.64 |
| CHEMBL1386141 | — | IC50 | = | 23601.0 | nM | 4.63 |
| CHEMBL1584538 | — | IC50 | = | 23622.0 | nM | 4.63 |
| CHEMBL1452812 | — | IC50 | = | 23831.0 | nM | 4.62 |
| CHEMBL1344766 | — | IC50 | = | 23970.0 | nM | 4.62 |