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Assay Detail

CHEMBL1614129

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Functional
PUBCHEM_BIOASSAY: Luminescence Cell-Based/Microorganism Primary HTS to Identify Inhibitors of Trypanosoma cruzi Infection. (Class of assay: confirmatory) [Related pubchem assays: 1885, 1968 ]
318
Total Activities
318
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Category confirmatory
Confidence 0 — Uncurated / Unknown
Curated By Autocuration

Target

Unchecked (CHEMBL612545)
Type UNCHECKED

Publication

PubChem BioAssay data set

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
EC50 318 7.14 8.40

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL1381971 1 8.40
CHEMBL1576088 1 8.22
CHEMBL536166 1 8.22
CHEMBL1610821 1 8.22
CHEMBL584442 1 8.22
CHEMBL1517801 1 8.15
CHEMBL530291 1 8.15
CHEMBL1716494 1 8.15
CHEMBL1378097 1 8.15
CHEMBL1468457 1 8.15
CHEMBL1516689 1 8.10
CHEMBL1525666 1 8.10
CHEMBL1583585 1 8.05
CHEMBL1406194 1 8.05
CHEMBL1425806 1 8.00
CHEMBL1379563 1 8.00
CHEMBL1473676 1 7.96
CHEMBL1415769 1 7.96
CHEMBL1307861 1 7.96
CHEMBL1613675 1 7.96
CHEMBL1472773 1 7.96
CHEMBL1588774 1 7.96
CHEMBL1413835 1 7.92
CHEMBL1421106 1 7.89
CHEMBL1359342 1 7.85
CHEMBL1557079 1 7.85
CHEMBL1518625 1 7.85
CHEMBL1450188 1 7.82
CHEMBL1454557 1 7.82
CHEMBL602759 1 7.82

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL1381971 EC50 = 4.0 nM 8.40
CHEMBL584442 EC50 = 6.0 nM 8.22
CHEMBL536166 EC50 = 6.0 nM 8.22
CHEMBL1610821 EC50 = 6.0 nM 8.22
CHEMBL1576088 EC50 = 6.0 nM 8.22
CHEMBL530291 EC50 = 7.0 nM 8.15
CHEMBL1517801 EC50 = 7.0 nM 8.15
CHEMBL1468457 EC50 = 7.0 nM 8.15
CHEMBL1716494 EC50 = 7.0 nM 8.15
CHEMBL1378097 EC50 = 7.0 nM 8.15
CHEMBL1525666 EC50 = 8.0 nM 8.10
CHEMBL1516689 EC50 = 8.0 nM 8.10
CHEMBL1406194 EC50 = 9.0 nM 8.05
CHEMBL1583585 EC50 = 9.0 nM 8.05
CHEMBL1425806 EC50 = 10.0 nM 8.00
CHEMBL1379563 EC50 = 10.0 nM 8.00
CHEMBL1307861 EC50 = 11.0 nM 7.96
CHEMBL1588774 EC50 = 11.0 nM 7.96
CHEMBL1473676 EC50 = 11.0 nM 7.96
CHEMBL1613675 EC50 = 11.0 nM 7.96
CHEMBL1415769 EC50 = 11.0 nM 7.96
CHEMBL1472773 EC50 = 11.0 nM 7.96
CHEMBL1413835 EC50 = 12.0 nM 7.92
CHEMBL1421106 EC50 = 13.0 nM 7.89
CHEMBL1557079 EC50 = 14.0 nM 7.85
CHEMBL1359342 EC50 = 14.0 nM 7.85
CHEMBL1518625 EC50 = 14.0 nM 7.85
CHEMBL1531377 EC50 = 15.0 nM 7.82
CHEMBL1450188 EC50 = 15.0 nM 7.82
CHEMBL602759 EC50 = 15.0 nM 7.82
CHEMBL1454557 EC50 = 15.0 nM 7.82
CHEMBL1327851 EC50 = 15.0 nM 7.82
CHEMBL1341517 EC50 = 16.0 nM 7.80
CHEMBL1385115 EC50 = 16.0 nM 7.80
CHEMBL1552445 EC50 = 16.0 nM 7.80
CHEMBL609628 EC50 = 17.0 nM 7.77
CHEMBL3197177 EC50 = 18.0 nM 7.75
CHEMBL1351537 EC50 = 19.0 nM 7.72
CHEMBL1536905 EC50 = 19.0 nM 7.72
CHEMBL3197634 EC50 = 19.0 nM 7.72
CHEMBL3190585 EC50 = 19.0 nM 7.72
CHEMBL1449336 EC50 = 19.0 nM 7.72
CHEMBL1457275 EC50 = 20.0 nM 7.70
CHEMBL1575081 EC50 = 20.0 nM 7.70
CHEMBL1564144 EC50 = 21.0 nM 7.68
CHEMBL1462215 EC50 = 21.0 nM 7.68
CHEMBL1417431 EC50 = 21.0 nM 7.68
CHEMBL609438 EC50 = 22.0 nM 7.66
CHEMBL1560237 EC50 = 22.0 nM 7.66
CHEMBL3214537 EC50 = 22.0 nM 7.66