Assay Detail
Functional
CHEMBL1614261
Review assay metadata, readout intent, target linkage, and publication context from the same page.
PUBCHEM_BIOASSAY: Luminescence Cell-Based/Microorganism Confirmation at Dose of Inhibitors of Trypanosoma cruzi Infection. (Class of assay: confirmatory) [Related pubchem assays: 1885, 1968 ]
25
Total Activities
25
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Category | confirmatory |
| Confidence | 0 — Uncurated / Unknown |
| Curated By | Autocuration |
Publication
PubChem BioAssay data set
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| EC50 | 25 | 6.47 | 7.66 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL1436964 | — | — | 1 | 7.66 |
| CHEMBL1382529 | — | — | 1 | 7.57 |
| CHEMBL1552445 | — | — | 1 | 7.50 |
| CHEMBL1459090 | — | — | 1 | 7.33 |
| CHEMBL1369986 | — | — | 1 | 7.24 |
| CHEMBL1372575 | — | — | 1 | 7.21 |
| CHEMBL1415084 | — | — | 1 | 7.17 |
| CHEMBL1331384 | — | — | 1 | 7.16 |
| CHEMBL1393939 | — | — | 1 | 7.01 |
| CHEMBL1474782 | — | — | 1 | 6.91 |
| CHEMBL1354193 | — | — | 1 | 6.75 |
| CHEMBL1328878 | — | — | 1 | 6.72 |
| CHEMBL1433324 | — | — | 1 | 6.64 |
| CHEMBL1332089 | — | — | 1 | 6.38 |
| CHEMBL1454008 | — | — | 1 | 6.22 |
| CHEMBL1411521 | — | — | 1 | 6.04 |
| CHEMBL1314621 | — | — | 1 | 6.04 |
| CHEMBL1441481 | — | — | 1 | 5.68 |
| CHEMBL1554427 | — | — | 1 | 5.66 |
| CHEMBL1593567 | — | — | 1 | 5.61 |
| CHEMBL1436871 | — | — | 1 | 5.60 |
| CHEMBL1444044 | — | — | 1 | 5.55 |
| CHEMBL1373415 | — | — | 1 | 5.51 |
| CHEMBL1515913 | — | — | 1 | 5.35 |
| CHEMBL1424146 | — | — | 1 | 5.14 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL1436964 | — | EC50 | = | 22.0 | nM | 7.66 |
| CHEMBL1382529 | — | EC50 | = | 27.0 | nM | 7.57 |
| CHEMBL1552445 | — | EC50 | = | 32.0 | nM | 7.50 |
| CHEMBL1459090 | — | EC50 | = | 47.0 | nM | 7.33 |
| CHEMBL1369986 | — | EC50 | = | 57.0 | nM | 7.24 |
| CHEMBL1372575 | — | EC50 | = | 62.0 | nM | 7.21 |
| CHEMBL1415084 | — | EC50 | = | 68.0 | nM | 7.17 |
| CHEMBL1331384 | — | EC50 | = | 69.0 | nM | 7.16 |
| CHEMBL1393939 | — | EC50 | = | 98.0 | nM | 7.01 |
| CHEMBL1474782 | — | EC50 | = | 123.0 | nM | 6.91 |
| CHEMBL1354193 | — | EC50 | = | 176.0 | nM | 6.75 |
| CHEMBL1328878 | — | EC50 | = | 192.0 | nM | 6.72 |
| CHEMBL1433324 | — | EC50 | = | 231.0 | nM | 6.64 |
| CHEMBL1332089 | — | EC50 | = | 417.0 | nM | 6.38 |
| CHEMBL1454008 | — | EC50 | = | 606.0 | nM | 6.22 |
| CHEMBL1411521 | — | EC50 | = | 903.0 | nM | 6.04 |
| CHEMBL1314621 | — | EC50 | = | 915.0 | nM | 6.04 |
| CHEMBL1441481 | — | EC50 | = | 2067.0 | nM | 5.68 |
| CHEMBL1554427 | — | EC50 | = | 2176.0 | nM | 5.66 |
| CHEMBL1593567 | — | EC50 | = | 2457.0 | nM | 5.61 |
| CHEMBL1436871 | — | EC50 | = | 2524.0 | nM | 5.60 |
| CHEMBL1444044 | — | EC50 | = | 2814.0 | nM | 5.55 |
| CHEMBL1373415 | — | EC50 | = | 3094.0 | nM | 5.51 |
| CHEMBL1515913 | — | EC50 | = | 4427.0 | nM | 5.35 |
| CHEMBL1424146 | — | EC50 | = | 7173.0 | nM | 5.14 |