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Assay Detail

CHEMBL1614412

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Functional
PUBCHEM_BIOASSAY: Dose Response Confirmation for DnaK Inhibitors. (Class of assay: confirmatory) [Related pubchem assays: 547 (Screening assay preceding this dose-response confirmation assay.)]
6
Total Activities
3
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Organism Escherichia coli str. K-12 substr. MG1655
Category confirmatory
Confidence 8 — Homologous single protein target
Curated By Autocuration

Target

Protein GrpE (CHEMBL1293284)
Type SINGLE PROTEIN
Organism Escherichia coli K-12

Publication

PubChem BioAssay data set

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 6 5.63 6.26

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL1365553 2 6.26
CHEMBL1256813 2 6.08
CHEMBL1256623 2 5.41

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL1365553 IC50 = 550.58 nM 6.26
CHEMBL1256813 IC50 = 837.09 nM 6.08
CHEMBL1256813 IC50 = 1624.86 nM 5.79
CHEMBL1365553 IC50 = 1664.33 nM 5.78
CHEMBL1256623 IC50 = 3921.72 nM 5.41
CHEMBL1256623 IC50 = 36310.06 nM 4.44