Assay Detail
Functional
CHEMBL1614418
Review assay metadata, readout intent, target linkage, and publication context from the same page.
PUBCHEM_BIOASSAY: In Vivo Angiogenesis Dose-Response Confirmation. (Class of assay: confirmatory) [Related pubchem assays: 732 (Assay preceding this confirmatory assay.)]
26
Total Activities
26
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Danio rerio |
| Category | confirmatory |
| Confidence | 1 — Organism |
| Curated By | Autocuration |
Publication
PubChem BioAssay data set
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 26 | 5.58 | 6.54 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL1481976 | — | — | 1 | 6.54 |
| CHEMBL126077 | INDIRUBIN-3-MONOXIME | — | 1 | 6.51 |
| CHEMBL1553033 | — | — | 1 | 6.46 |
| CHEMBL1077291 | — | — | 1 | 6.42 |
| CHEMBL1450830 | — | — | 1 | 6.28 |
| CHEMBL1597388 | — | — | 1 | 6.17 |
| CHEMBL23330 | TRETAZICAR | 2.0 | 1 | 5.92 |
| CHEMBL1589857 | — | — | 1 | 5.91 |
| CHEMBL367345 | — | — | 1 | 5.66 |
| CHEMBL1597016 | — | — | 1 | 5.60 |
| CHEMBL1364560 | — | — | 1 | 5.48 |
| CHEMBL1613176 | — | — | 1 | 5.40 |
| CHEMBL1444075 | — | — | 1 | 5.37 |
| CHEMBL543876 | — | — | 1 | 5.24 |
| CHEMBL1315255 | — | — | 1 | 5.20 |
| CHEMBL415879 | PHENANTHROLINE | — | 1 | 5.12 |
| CHEMBL1480 | FELODIPINE | 4.0 | 1 | 5.04 |
| CHEMBL7917 | TYRPHOSTIN AG-1478 | — | 1 | 4.90 |
| CHEMBL1515403 | — | — | 1 | 4.88 |
| CHEMBL85139 | RUTAECARPINE | — | 1 | 4.59 |
| CHEMBL1255831 | E1001 | — | 1 | 4.50 |
| CHEMBL328710 | — | — | 1 | - |
| CHEMBL1394987 | — | — | 1 | - |
| CHEMBL1496938 | — | — | 1 | - |
| CHEMBL1276127 | INDIRUBIN | 2.0 | 1 | - |
| CHEMBL1314295 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL1481976 | — | IC50 | = | 290.0 | nM | 6.54 |
| CHEMBL126077 | INDIRUBIN-3-MONOXIME | IC50 | = | 310.0 | nM | 6.51 |
| CHEMBL1553033 | — | IC50 | = | 350.0 | nM | 6.46 |
| CHEMBL1077291 | — | IC50 | = | 380.0 | nM | 6.42 |
| CHEMBL1450830 | — | IC50 | = | 520.0 | nM | 6.28 |
| CHEMBL1597388 | — | IC50 | = | 680.0 | nM | 6.17 |
| CHEMBL23330 | TRETAZICAR | IC50 | = | 1200.0 | nM | 5.92 |
| CHEMBL1589857 | — | IC50 | = | 1230.0 | nM | 5.91 |
| CHEMBL367345 | — | IC50 | = | 2170.0 | nM | 5.66 |
| CHEMBL1597016 | — | IC50 | = | 2500.0 | nM | 5.60 |
| CHEMBL1364560 | — | IC50 | = | 3280.0 | nM | 5.48 |
| CHEMBL1613176 | — | IC50 | = | 4010.0 | nM | 5.40 |
| CHEMBL1444075 | — | IC50 | = | 4240.0 | nM | 5.37 |
| CHEMBL543876 | — | IC50 | = | 5730.0 | nM | 5.24 |
| CHEMBL1315255 | — | IC50 | = | 6320.0 | nM | 5.20 |
| CHEMBL415879 | PHENANTHROLINE | IC50 | = | 7510.0 | nM | 5.12 |
| CHEMBL1480 | FELODIPINE | IC50 | = | 9210.0 | nM | 5.04 |
| CHEMBL7917 | TYRPHOSTIN AG-1478 | IC50 | = | 12660.0 | nM | 4.90 |
| CHEMBL1515403 | — | IC50 | = | 13140.0 | nM | 4.88 |
| CHEMBL85139 | RUTAECARPINE | IC50 | = | 25490.0 | nM | 4.59 |
| CHEMBL1255831 | E1001 | IC50 | = | 31620.0 | nM | 4.50 |
| CHEMBL328710 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL1394987 | — | IC50 | < | 300.0 | nM | - |
| CHEMBL1496938 | — | IC50 | > | 10000.0 | nM | - |
| CHEMBL1276127 | INDIRUBIN | IC50 | < | 100.0 | nM | - |
| CHEMBL1314295 | — | IC50 | > | 30000.0 | nM | - |