Assay Detail
Functional
CHEMBL1614480
Review assay metadata, readout intent, target linkage, and publication context from the same page.
PUBCHEM_BIOASSAY: HTS Dose response counterscreen for assays utilizing the enzyme, b-galactosidase. (Class of assay: confirmatory) [Related pubchem assays (depositor defined):AID1777, AID1778, AID1785, AID1786, AID2284, AID2285, AID2348, AID2352, AID2357, AID2359, AID2370, AID2420, AID2478, AID2491, AID2492, AID2493, AID2495, AID2497, AID2498, AID2500, AID434981, AID449737, AID463105, AID485352, AID488822, AID488842, AID488935]
211
Total Activities
211
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Escherichia coli |
| Category | confirmatory |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
PubChem BioAssay data set
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| EC50 | 211 | 4.89 | 5.78 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL1973773 | — | — | 1 | 5.78 |
| CHEMBL1442698 | — | — | 1 | 5.52 |
| CHEMBL1300269 | — | — | 1 | 5.50 |
| CHEMBL1598011 | — | — | 1 | 5.10 |
| CHEMBL1565646 | — | — | 1 | 5.05 |
| CHEMBL1306723 | — | — | 1 | 5.04 |
| CHEMBL1605583 | — | — | 1 | 5.01 |
| CHEMBL1606916 | — | — | 1 | 4.99 |
| CHEMBL1462003 | — | — | 1 | 4.95 |
| CHEMBL1384246 | — | — | 1 | 4.94 |
| CHEMBL1548770 | — | — | 1 | 4.88 |
| CHEMBL1302391 | — | — | 1 | 4.85 |
| CHEMBL1557816 | — | — | 1 | 4.85 |
| CHEMBL1433128 | — | — | 1 | 4.84 |
| CHEMBL1311879 | — | — | 1 | 4.84 |
| CHEMBL1529511 | — | — | 1 | 4.83 |
| CHEMBL1456232 | — | — | 1 | 4.83 |
| CHEMBL1596609 | — | — | 1 | 4.78 |
| CHEMBL1477640 | — | — | 1 | 4.76 |
| CHEMBL1522851 | — | — | 1 | 4.74 |
| CHEMBL1586491 | — | — | 1 | 4.69 |
| CHEMBL1350780 | — | — | 1 | 4.66 |
| CHEMBL1311826 | — | — | 1 | 4.63 |
| CHEMBL1495714 | — | — | 1 | 4.62 |
| CHEMBL1447284 | — | — | 1 | 4.61 |
| CHEMBL1539624 | — | — | 1 | 4.60 |
| CHEMBL1400298 | — | — | 1 | 4.59 |
| CHEMBL1422078 | — | — | 1 | 4.52 |
| CHEMBL1976317 | — | — | 1 | - |
| CHEMBL1554920 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL1973773 | — | EC50 | = | 1665.0 | nM | 5.78 |
| CHEMBL1442698 | — | EC50 | = | 3025.0 | nM | 5.52 |
| CHEMBL1300269 | — | EC50 | = | 3160.0 | nM | 5.50 |
| CHEMBL1598011 | — | EC50 | = | 7925.0 | nM | 5.10 |
| CHEMBL1565646 | — | EC50 | = | 8915.0 | nM | 5.05 |
| CHEMBL1306723 | — | EC50 | = | 9225.0 | nM | 5.04 |
| CHEMBL1605583 | — | EC50 | = | 9665.0 | nM | 5.01 |
| CHEMBL1606916 | — | EC50 | = | 10295.0 | nM | 4.99 |
| CHEMBL1462003 | — | EC50 | = | 11300.0 | nM | 4.95 |
| CHEMBL1384246 | — | EC50 | = | 11500.0 | nM | 4.94 |
| CHEMBL1548770 | — | EC50 | = | 13050.0 | nM | 4.88 |
| CHEMBL1302391 | — | EC50 | = | 14150.0 | nM | 4.85 |
| CHEMBL1557816 | — | EC50 | = | 14100.0 | nM | 4.85 |
| CHEMBL1433128 | — | EC50 | = | 14350.0 | nM | 4.84 |
| CHEMBL1311879 | — | EC50 | = | 14500.0 | nM | 4.84 |
| CHEMBL1529511 | — | EC50 | = | 14750.0 | nM | 4.83 |
| CHEMBL1456232 | — | EC50 | = | 14650.0 | nM | 4.83 |
| CHEMBL1596609 | — | EC50 | = | 16650.0 | nM | 4.78 |
| CHEMBL1477640 | — | EC50 | = | 17450.0 | nM | 4.76 |
| CHEMBL1522851 | — | EC50 | = | 18150.0 | nM | 4.74 |
| CHEMBL1586491 | — | EC50 | = | 20350.0 | nM | 4.69 |
| CHEMBL1350780 | — | EC50 | = | 21950.0 | nM | 4.66 |
| CHEMBL1311826 | — | EC50 | = | 23550.0 | nM | 4.63 |
| CHEMBL1495714 | — | EC50 | = | 23850.0 | nM | 4.62 |
| CHEMBL1447284 | — | EC50 | = | 24550.0 | nM | 4.61 |
| CHEMBL1539624 | — | EC50 | = | 25300.0 | nM | 4.60 |
| CHEMBL1400298 | — | EC50 | = | 25700.0 | nM | 4.59 |
| CHEMBL1422078 | — | EC50 | = | 30100.0 | nM | 4.52 |
| CHEMBL1585390 | — | EC50 | > | 31500.0 | nM | - |
| CHEMBL1455045 | — | EC50 | > | 31500.0 | nM | - |
| CHEMBL1609419 | — | EC50 | > | 31500.0 | nM | - |
| CHEMBL3197021 | — | EC50 | > | 31500.0 | nM | - |
| CHEMBL1964873 | — | EC50 | > | 31500.0 | nM | - |
| CHEMBL1301723 | — | EC50 | > | 31500.0 | nM | - |
| CHEMBL1417204 | — | EC50 | > | 31500.0 | nM | - |
| CHEMBL1504142 | — | EC50 | > | 31500.0 | nM | - |
| CHEMBL428064 | — | EC50 | > | 31500.0 | nM | - |
| CHEMBL1718 | NALOXONE HYDROCHLORIDE | EC50 | > | 31500.0 | nM | - |
| CHEMBL1428935 | — | EC50 | > | 31500.0 | nM | - |
| CHEMBL1416089 | — | EC50 | > | 31500.0 | nM | - |
| CHEMBL1460705 | — | EC50 | > | 31500.0 | nM | - |
| CHEMBL140425 | — | EC50 | > | 31500.0 | nM | - |
| CHEMBL1442120 | — | EC50 | > | 31500.0 | nM | - |
| CHEMBL1423597 | — | EC50 | > | 31500.0 | nM | - |
| CHEMBL1603353 | — | EC50 | > | 31500.0 | nM | - |
| CHEMBL1455427 | — | EC50 | > | 31500.0 | nM | - |
| CHEMBL1558590 | — | EC50 | > | 31500.0 | nM | - |
| CHEMBL1384726 | — | EC50 | > | 31500.0 | nM | - |
| CHEMBL1319867 | — | EC50 | > | 31500.0 | nM | - |
| CHEMBL1553074 | — | EC50 | > | 31500.0 | nM | - |