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Assay Detail

CHEMBL1636227

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Functional
Antiviral activity against GCV-resistant Human cytomegalovirus 759rD100 harboring 4-aa deletion (638-641) in UL97 kinase and DNA polymerase A987G mutant infected in human foreskin fibroblast by plaque reduction assay
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Organism Human betaherpesvirus 5
Confidence 1 — Organism
Curated By Autocuration

Target

Human betaherpesvirus 5 (CHEMBL371)
Type ORGANISM
Organism Human betaherpesvirus 5

Publication

A 6-aminoquinolone compound, WC5, with potent and selective anti-human cytomegalovirus activity.
Mercorelli B, Muratore G, Sinigalia E, Tabarrini O, Biasolo MA, Cecchetti V, Palù G, Loregian A.
Antimicrob Agents Chemother (2009) 53 : 312 -315
PubMed 19015358 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
EC50 1 6.05 6.05

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL127498 1 6.05

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL127498 EC50 = 900.0 nM 6.05