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Assay Detail

CHEMBL1637305

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Functional
Antiviral activity against at 0.3 MOI Dengue virus 2 infected in human A549 cells assessed as level of E protein after 48 hrs by ELISA
11
Total Activities
11
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Organism dengue virus type 2
Cell Type A549
Confidence 1 — Organism
Curated By Autocuration

Target

dengue virus type 2 (CHEMBL613966)
Type ORGANISM
Organism dengue virus type 2

Publication

Inhibition of dengue virus RNA synthesis by an adenosine nucleoside.
Chen YL, Yin Z, Duraiswamy J, Schul W, Lim CC, Liu B, Xu HY, Qing M, Yip A, Wang G, Chan WL, Tan HP, Lo M, Liung S, Kondreddi RR, Rao R, Gu H, He H, Keller TH, Shi PY.
Antimicrob Agents Chemother (2010) 54 : 2932 -2939
PubMed 20457821 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
EC50 11 5.93 6.38

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL1631768 1 6.38
CHEMBL1630221 1 6.16
CHEMBL73809 1 5.95
CHEMBL1631698 1 5.85
CHEMBL1630219 1 5.70
CHEMBL1631769 1 5.51
CHEMBL311635 1 -
CHEMBL1631697 1 -
CHEMBL1631699 1 -
CHEMBL98778 2'-ETHYNYL-D-CYTIDINE 1 -
CHEMBL1631700 1 -

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL1631768 EC50 = 420.0 nM 6.38
CHEMBL1630221 EC50 = 700.0 nM 6.16
CHEMBL73809 EC50 = 1120.0 nM 5.95
CHEMBL1631698 EC50 = 1410.0 nM 5.85
CHEMBL1630219 EC50 = 2000.0 nM 5.70
CHEMBL1631769 EC50 = 3100.0 nM 5.51
CHEMBL311635 EC50 > 100000.0 nM -
CHEMBL1631697 EC50 > 50000.0 nM -
CHEMBL1631699 EC50 > 100000.0 nM -
CHEMBL98778 2'-ETHYNYL-D-CYTIDINE EC50 > 100000.0 nM -
CHEMBL1631700 EC50 > 100000.0 nM -