Assay Detail
Binding
CHEMBL1639355
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Inhibition of human Chymase
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
2-Azetidinone--a new profile of various pharmacological activities.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 2 | 8.93 | 9.34 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL1631751 | — | — | 1 | 9.34 |
| CHEMBL1631756 | — | — | 1 | 8.51 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL1631751 | — | IC50 | = | 0.46 | nM | 9.34 |
| CHEMBL1631756 | — | IC50 | = | 3.1 | nM | 8.51 |