Assay Detail
Binding
CHEMBL1647731
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Inhibition of calmodulin assessed as inhibition of calmodulin-calcium-PDE1 complex formation
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Confidence | 8 — Homologous single protein target |
| Curated By | Autocuration |
Publication
Vasorelaxant effect of flavonoids through calmodulin inhibition: Ex vivo, in vitro, and in silico approaches.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 1 | 4.13 | 4.13 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL449317 | HESPERIDIN | 3.0 | 1 | 4.13 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL449317 | HESPERIDIN | IC50 | = | 74000.0 | nM | 4.13 |