Assay Detail
Binding
CHEMBL1664438
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Inhibition of recombinant anthrax lethal factor after 30 mins by fluorescence assay
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Bacillus anthracis |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
Identifying chelators for metalloprotein inhibitors using a fragment-based approach.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 2 | 3.69 | 3.69 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL1649594 | — | — | 1 | 3.69 |
| CHEMBL734 | ACETOHYDROXAMIC ACID | 4.0 | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL1649594 | — | IC50 | = | 204000.0 | nM | 3.69 |
| CHEMBL734 | ACETOHYDROXAMIC ACID | IC50 | = | 11400000.0 | nM | - |