Assay Detail
Functional
CHEMBL1680809
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Antagonist activity against rat P2X4 receptor expressed in Xenopus laevis oocyte assessed as inhibition of alpha, beta-meATP-induced inward current by two-electrode voltage-clamp electrophysiology
62
Total Activities
62
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Rattus norvegicus |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
Discovery of potent competitive antagonists and positive modulators of the P2X2 receptor.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 62 | 4.40 | 4.40 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL134193 | CIBACRON BLUE 3GA | — | 1 | 4.40 |
| CHEMBL597591 | — | — | 1 | - |
| CHEMBL1672107 | — | — | 1 | - |
| CHEMBL1672106 | — | — | 1 | - |
| CHEMBL509572 | — | — | 1 | - |
| CHEMBL1672105 | — | — | 1 | - |
| CHEMBL496229 | — | — | 1 | - |
| CHEMBL496401 | — | — | 1 | - |
| CHEMBL499580 | — | — | 1 | - |
| CHEMBL499428 | — | — | 1 | - |
| CHEMBL131271 | — | — | 1 | - |
| CHEMBL1672104 | — | — | 1 | - |
| CHEMBL455536 | — | — | 1 | - |
| CHEMBL1672103 | — | — | 1 | - |
| CHEMBL450832 | — | — | 1 | - |
| CHEMBL596982 | — | — | 1 | - |
| CHEMBL1672101 | — | — | 1 | - |
| CHEMBL1672100 | — | — | 1 | - |
| CHEMBL495796 | — | — | 1 | - |
| CHEMBL133576 | ACID BLUE 129 | — | 1 | - |
| CHEMBL498038 | — | — | 1 | - |
| CHEMBL495834 | — | — | 1 | - |
| CHEMBL521709 | — | — | 1 | - |
| CHEMBL522053 | — | — | 1 | - |
| CHEMBL524284 | — | — | 1 | - |
| CHEMBL404659 | — | — | 1 | - |
| CHEMBL271688 | — | — | 1 | - |
| CHEMBL496012 | — | — | 1 | - |
| CHEMBL597820 | — | — | 1 | - |
| CHEMBL1672102 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL134193 | CIBACRON BLUE 3GA | IC50 | = | 40000.0 | nM | 4.40 |
| CHEMBL445413 | — | IC50 | > | 10000.0 | nM | - |
| CHEMBL1672105 | — | IC50 | - | — | - | |
| CHEMBL509572 | — | IC50 | > | 10000.0 | nM | - |
| CHEMBL1672106 | — | IC50 | > | 10000.0 | nM | - |
| CHEMBL1672107 | — | IC50 | - | — | - | |
| CHEMBL223344 | RB 2 | IC50 | - | — | - | |
| CHEMBL1671995 | — | IC50 | > | 10000.0 | nM | - |
| CHEMBL596985 | — | IC50 | > | 10000.0 | nM | - |
| CHEMBL1671991 | — | IC50 | > | 10000.0 | nM | - |
| CHEMBL606414 | — | IC50 | > | 10000.0 | nM | - |
| CHEMBL498423 | — | IC50 | > | 10000.0 | nM | - |
| CHEMBL256864 | — | IC50 | > | 10000.0 | nM | - |
| CHEMBL496229 | — | IC50 | > | 10000.0 | nM | - |
| CHEMBL404450 | — | IC50 | > | 10000.0 | nM | - |
| CHEMBL1671992 | — | IC50 | - | — | - | |
| CHEMBL1671993 | — | IC50 | - | — | - | |
| CHEMBL402239 | — | IC50 | > | 10000.0 | nM | - |
| CHEMBL256688 | — | IC50 | > | 10000.0 | nM | - |
| CHEMBL1671994 | — | IC50 | - | — | - | |
| CHEMBL522725 | — | IC50 | > | 10000.0 | nM | - |
| CHEMBL496030 | — | IC50 | > | 10000.0 | nM | - |
| CHEMBL257495 | — | IC50 | > | 10000.0 | nM | - |
| CHEMBL256057 | ACID BLUE 25 | IC50 | > | 10000.0 | nM | - |
| CHEMBL401735 | — | IC50 | > | 10000.0 | nM | - |
| CHEMBL1671996 | — | IC50 | - | — | - | |
| CHEMBL495796 | — | IC50 | > | 10000.0 | nM | - |
| CHEMBL1672102 | — | IC50 | > | 10000.0 | nM | - |
| CHEMBL597820 | — | IC50 | > | 10000.0 | nM | - |
| CHEMBL496012 | — | IC50 | > | 10000.0 | nM | - |
| CHEMBL271688 | — | IC50 | > | 10000.0 | nM | - |
| CHEMBL404659 | — | IC50 | - | — | - | |
| CHEMBL524284 | — | IC50 | > | 10000.0 | nM | - |
| CHEMBL522053 | — | IC50 | > | 10000.0 | nM | - |
| CHEMBL521709 | — | IC50 | > | 10000.0 | nM | - |
| CHEMBL495834 | — | IC50 | > | 10000.0 | nM | - |
| CHEMBL498038 | — | IC50 | > | 10000.0 | nM | - |
| CHEMBL133576 | ACID BLUE 129 | IC50 | > | 10000.0 | nM | - |
| CHEMBL496401 | — | IC50 | > | 10000.0 | nM | - |
| CHEMBL1672100 | — | IC50 | - | — | - | |
| CHEMBL1672101 | — | IC50 | - | — | - | |
| CHEMBL597591 | — | IC50 | > | 10000.0 | nM | - |
| CHEMBL596982 | — | IC50 | > | 10000.0 | nM | - |
| CHEMBL450832 | — | IC50 | > | 10000.0 | nM | - |
| CHEMBL1672103 | — | IC50 | > | 10000.0 | nM | - |
| CHEMBL455536 | — | IC50 | - | — | - | |
| CHEMBL1672104 | — | IC50 | > | 10000.0 | nM | - |
| CHEMBL131271 | — | IC50 | > | 10000.0 | nM | - |
| CHEMBL499428 | — | IC50 | > | 10000.0 | nM | - |
| CHEMBL499580 | — | IC50 | > | 10000.0 | nM | - |