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Assay Detail

CHEMBL1681017

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Functional
Antiparasitic activity against Leishmania infantum MHOM/ES/1993/BCN-99 after 3 days by Alamar blue assay
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Organism Leishmania infantum
Confidence 1 — Organism
Curated By Autocuration

Target

Leishmania infantum (CHEMBL612848)
Type ORGANISM
Organism Leishmania infantum

Publication

Sitamaquine sensitivity in Leishmania species is not mediated by drug accumulation in acidocalcisomes.
López-Martín C, Pérez-Victoria JM, Carvalho L, Castanys S, Gamarro F.
Antimicrob Agents Chemother (2008) 52 : 4030 -4036
PubMed 18794384 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
EC50 1 5.02 5.02

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL3142235 1 5.02

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL3142235 EC50 = 9500.0 nM 5.02