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Assay Detail

CHEMBL1685195

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Functional
Antagonist activity at CXCR4 in human CEM-CCRF cells assessed as inhibition of SDF-1-induced calcium signaling
22
Total Activities
22
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Organism Homo sapiens
Cell Type CEM-CCRF
Confidence 9 — Direct single protein target
Curated By Autocuration

Target

C-X-C chemokine receptor type 4 (CHEMBL2107)
Type SINGLE PROTEIN
Organism Homo sapiens

Publication

Design of novel CXCR4 antagonists that are potent inhibitors of T-tropic (X4) HIV-1 replication.
Skerlj R, Bridger G, McEachern E, Harwig C, Smith C, Kaller A, Veale D, Yee H, Skupinska K, Wauthy R, Wang L, Baird I, Zhu Y, Burrage K, Yang W, Sartori M, Huskens D, De Clercq E, Schols D.
Bioorg Med Chem Lett (2011) 21 : 1414 -1418
PubMed 21295470 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 22 7.28 8.10

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL1682993 1 8.10
CHEMBL1682854 1 7.75
CHEMBL1682989 1 7.75
CHEMBL1682859 1 7.72
CHEMBL1682992 1 7.70
CHEMBL1682986 1 7.64
CHEMBL1682863 1 7.57
CHEMBL1682856 1 7.46
CHEMBL1682858 1 7.42
CHEMBL1682866 1 7.36
CHEMBL1682860 1 7.31
CHEMBL1682857 1 7.28
CHEMBL1682864 1 7.20
CHEMBL1682990 1 7.18
CHEMBL1682987 1 7.14
CHEMBL1099015 1 7.13
CHEMBL1682865 1 7.10
CHEMBL1682855 1 7.04
CHEMBL1682988 1 6.96
CHEMBL1682862 1 6.89
CHEMBL1682991 1 6.74
CHEMBL1682861 1 5.79

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL1682993 IC50 = 8.0 nM 8.10
CHEMBL1682854 IC50 = 18.0 nM 7.75
CHEMBL1682989 IC50 = 18.0 nM 7.75
CHEMBL1682859 IC50 = 19.0 nM 7.72
CHEMBL1682992 IC50 = 20.0 nM 7.70
CHEMBL1682986 IC50 = 23.0 nM 7.64
CHEMBL1682863 IC50 = 27.0 nM 7.57
CHEMBL1682856 IC50 = 35.0 nM 7.46
CHEMBL1682858 IC50 = 38.0 nM 7.42
CHEMBL1682866 IC50 = 44.0 nM 7.36
CHEMBL1682860 IC50 = 49.0 nM 7.31
CHEMBL1682857 IC50 = 53.0 nM 7.28
CHEMBL1682864 IC50 = 63.0 nM 7.20
CHEMBL1682990 IC50 = 66.0 nM 7.18
CHEMBL1682987 IC50 = 72.0 nM 7.14
CHEMBL1099015 IC50 = 74.0 nM 7.13
CHEMBL1682865 IC50 = 79.0 nM 7.10
CHEMBL1682855 IC50 = 91.0 nM 7.04
CHEMBL1682988 IC50 = 111.0 nM 6.96
CHEMBL1682862 IC50 = 129.0 nM 6.89
CHEMBL1682991 IC50 = 183.0 nM 6.74
CHEMBL1682861 IC50 = 1621.0 nM 5.79