Assay Detail
Binding
CHEMBL1693308
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Inhibition of Pdr5p-dependent UTPase activity in Saccharomyces cerevisiae AD124567 assessed as release of inorganic phosphate after 60 mins by Lineweaver-Burk plot
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Saccharomyces cerevisiae |
| Confidence | 0 — Uncurated / Unknown |
| Curated By | Autocuration |
Publication
Oroidin inhibits the activity of the multidrug resistance target Pdr5p from yeast plasma membranes.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 1 | 4.89 | 4.89 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL397591 | OROIDIN | — | 1 | 4.89 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL397591 | OROIDIN | IC50 | = | 13000.0 | nM | 4.89 |