Assay Detail
Binding
CHEMBL1696445
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Activation of rat AMPK after 15 mins
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Rattus norvegicus |
| Confidence | 0 — Uncurated / Unknown |
| Curated By | Autocuration |
Publication
A Potent and Selective AMPK Activator That Inhibits de Novo Lipogenesis.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| EC50 | 2 | 5.88 | 7.68 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL1688230 | — | — | 1 | 7.68 |
| CHEMBL483849 | — | — | 1 | 4.08 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL1688230 | — | EC50 | = | 21.0 | nM | 7.68 |
| CHEMBL483849 | — | EC50 | = | 84000.0 | nM | 4.08 |