Assay Detail
Functional
CHEMBL1737897
Review assay metadata, readout intent, target linkage, and publication context from the same page.
PUBCHEM_BIOASSAY: Counterscreen for antagonists of the orexin 1 receptor (OX1R; HCRTR1): Homogeneous time resolved fluorescence (HTRF)-based cell-based dose response assay to identify antagonists of the parental CHO-K1 cell line. (Class of assay: confirmatory) [Related pubchem assays (depositor defined):AID434989, AID435008, AID463079, AID485270, AID492963, AID492964, AID492965, AID493232, AID504699, AID504701]
247
Total Activities
247
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Cricetulus griseus |
| Cell Type | CHO-K1 |
| Category | confirmatory |
| Confidence | 1 — Organism |
| Curated By | Autocuration |
Publication
PubChem BioAssay data set
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 247 | 4.49 | 4.98 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL1375038 | — | — | 1 | 4.98 |
| CHEMBL1367399 | — | — | 1 | 4.93 |
| CHEMBL1466856 | — | — | 1 | 4.73 |
| CHEMBL1595403 | — | — | 1 | 4.57 |
| CHEMBL1336039 | — | — | 1 | 4.52 |
| CHEMBL1512619 | — | — | 1 | 4.47 |
| CHEMBL1516768 | — | — | 1 | 4.46 |
| CHEMBL1532403 | — | — | 1 | 4.39 |
| CHEMBL1995997 | — | — | 1 | 4.33 |
| CHEMBL1533279 | — | — | 1 | 4.29 |
| CHEMBL1964878 | — | — | 1 | 4.27 |
| CHEMBL1572480 | — | — | 1 | 4.25 |
| CHEMBL1518566 | — | — | 1 | 4.21 |
| CHEMBL1699081 | — | — | 1 | - |
| CHEMBL1571574 | — | — | 1 | - |
| CHEMBL1458435 | — | — | 1 | - |
| CHEMBL1465216 | — | — | 1 | - |
| CHEMBL1379934 | — | — | 1 | - |
| CHEMBL1576843 | — | — | 1 | - |
| CHEMBL1493516 | — | — | 1 | - |
| CHEMBL1334210 | — | — | 1 | - |
| CHEMBL1481716 | — | — | 1 | - |
| CHEMBL1977808 | — | — | 1 | - |
| CHEMBL1378896 | — | — | 1 | - |
| CHEMBL1384723 | — | — | 1 | - |
| CHEMBL1977763 | — | — | 1 | - |
| CHEMBL1364699 | — | — | 1 | - |
| CHEMBL1491556 | — | — | 1 | - |
| CHEMBL1333250 | — | — | 1 | - |
| CHEMBL1448743 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL1375038 | — | IC50 | = | 10504.0 | nM | 4.98 |
| CHEMBL1367399 | — | IC50 | = | 11606.0 | nM | 4.93 |
| CHEMBL1466856 | — | IC50 | = | 18528.0 | nM | 4.73 |
| CHEMBL1595403 | — | IC50 | = | 27031.0 | nM | 4.57 |
| CHEMBL1336039 | — | IC50 | = | 29946.0 | nM | 4.52 |
| CHEMBL1512619 | — | IC50 | = | 33555.0 | nM | 4.47 |
| CHEMBL1516768 | — | IC50 | = | 35039.0 | nM | 4.46 |
| CHEMBL1532403 | — | IC50 | = | 40654.0 | nM | 4.39 |
| CHEMBL1995997 | — | IC50 | = | 46826.0 | nM | 4.33 |
| CHEMBL1533279 | — | IC50 | = | 50660.0 | nM | 4.29 |
| CHEMBL1964878 | — | IC50 | = | 53660.0 | nM | 4.27 |
| CHEMBL1572480 | — | IC50 | = | 56925.0 | nM | 4.25 |
| CHEMBL1518566 | — | IC50 | = | 62048.0 | nM | 4.21 |
| CHEMBL1581581 | — | IC50 | > | 66172.0 | nM | - |
| CHEMBL1307031 | — | IC50 | > | 66191.0 | nM | - |
| CHEMBL1520702 | — | IC50 | > | 66258.0 | nM | - |
| CHEMBL1721971 | — | IC50 | > | 66174.0 | nM | - |
| CHEMBL1327720 | — | IC50 | > | 66238.0 | nM | - |
| CHEMBL1440341 | — | IC50 | > | 66205.0 | nM | - |
| CHEMBL1501678 | — | IC50 | > | 66207.0 | nM | - |
| CHEMBL1363571 | — | IC50 | > | 66209.0 | nM | - |
| CHEMBL1612190 | — | IC50 | > | 66225.0 | nM | - |
| CHEMBL1590005 | — | IC50 | > | 66232.0 | nM | - |
| CHEMBL1528787 | — | IC50 | > | 66225.0 | nM | - |
| CHEMBL1342888 | — | IC50 | > | 66232.0 | nM | - |
| CHEMBL1560993 | — | IC50 | > | 66168.0 | nM | - |
| CHEMBL1714761 | — | IC50 | > | 66211.0 | nM | - |
| CHEMBL2006840 | — | IC50 | > | 66225.0 | nM | - |
| CHEMBL1502109 | — | IC50 | > | 66232.0 | nM | - |
| CHEMBL1514800 | — | IC50 | > | 66278.0 | nM | - |
| CHEMBL1518032 | — | IC50 | > | 66232.0 | nM | - |
| CHEMBL1496820 | — | IC50 | > | 66298.0 | nM | - |
| CHEMBL1540815 | — | IC50 | > | 66223.0 | nM | - |
| CHEMBL1430677 | — | IC50 | > | 66209.0 | nM | - |
| CHEMBL1343392 | — | IC50 | > | 66221.0 | nM | - |
| CHEMBL1480014 | — | IC50 | > | 66215.0 | nM | - |
| CHEMBL1521046 | — | IC50 | > | 66168.0 | nM | - |
| CHEMBL1562279 | — | IC50 | > | 66218.0 | nM | - |
| CHEMBL1369963 | — | IC50 | > | 66272.0 | nM | - |
| CHEMBL1546895 | — | IC50 | > | 66211.0 | nM | - |
| CHEMBL1967103 | — | IC50 | > | 66232.0 | nM | - |
| CHEMBL1365949 | — | IC50 | > | 66224.0 | nM | - |
| CHEMBL1988282 | — | IC50 | > | 66222.0 | nM | - |
| CHEMBL1355104 | — | IC50 | > | 66197.0 | nM | - |
| CHEMBL1733477 | — | IC50 | > | 66172.0 | nM | - |
| CHEMBL1716146 | — | IC50 | > | 66177.0 | nM | - |
| CHEMBL2004183 | — | IC50 | > | 66225.0 | nM | - |
| CHEMBL1386871 | — | IC50 | > | 66265.0 | nM | - |
| CHEMBL1604928 | — | IC50 | > | 66211.0 | nM | - |
| CHEMBL1970286 | — | IC50 | > | 66232.0 | nM | - |