Assay Detail
Functional
CHEMBL1737962
Review assay metadata, readout intent, target linkage, and publication context from the same page.
PUBCHEM_BIOASSAY: SAR selectivity analysis of spectral interference of small molecule detect in Homogeneous Time-Resolved Fluorescence Resonance Energy Transfer (HTRF). (Class of assay: confirmatory) [Related pubchem assays (depositor defined):AID2073, AID2091, AID2093]
28
Total Activities
28
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Category | confirmatory |
| Confidence | 0 — Uncurated / Unknown |
| Curated By | Autocuration |
Publication
PubChem BioAssay data set
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 28 | 5.04 | 5.54 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL1486729 | — | — | 1 | 5.54 |
| CHEMBL1546396 | — | — | 1 | 5.53 |
| CHEMBL1526690 | — | — | 1 | 5.38 |
| CHEMBL1467976 | — | — | 1 | 5.35 |
| CHEMBL1530272 | — | — | 1 | 5.25 |
| CHEMBL1719095 | — | — | 1 | 5.18 |
| CHEMBL1707169 | — | — | 1 | 5.13 |
| CHEMBL1587502 | — | — | 1 | 5.05 |
| CHEMBL1457149 | — | — | 1 | 4.89 |
| CHEMBL1700951 | — | — | 1 | 4.82 |
| CHEMBL1530437 | — | — | 1 | 4.79 |
| CHEMBL1535613 | — | — | 1 | 4.70 |
| CHEMBL1399979 | — | — | 1 | 4.58 |
| CHEMBL1402286 | — | — | 1 | 4.43 |
| CHEMBL1494713 | — | — | 1 | - |
| CHEMBL1585333 | — | — | 1 | - |
| CHEMBL1399577 | — | — | 1 | - |
| CHEMBL1334484 | — | — | 1 | - |
| CHEMBL1426689 | — | — | 1 | - |
| CHEMBL1507308 | — | — | 1 | - |
| CHEMBL1328773 | — | — | 1 | - |
| CHEMBL1310699 | — | — | 1 | - |
| CHEMBL1481413 | — | — | 1 | - |
| CHEMBL1446655 | — | — | 1 | - |
| CHEMBL1600114 | — | — | 1 | - |
| CHEMBL1404231 | — | — | 1 | - |
| CHEMBL1383746 | — | — | 1 | - |
| CHEMBL1548870 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL1486729 | — | IC50 | = | 2861.0 | nM | 5.54 |
| CHEMBL1546396 | — | IC50 | = | 2981.0 | nM | 5.53 |
| CHEMBL1526690 | — | IC50 | = | 4142.0 | nM | 5.38 |
| CHEMBL1467976 | — | IC50 | = | 4421.0 | nM | 5.35 |
| CHEMBL1530272 | — | IC50 | = | 5591.0 | nM | 5.25 |
| CHEMBL1719095 | — | IC50 | = | 6550.0 | nM | 5.18 |
| CHEMBL1707169 | — | IC50 | = | 7323.0 | nM | 5.13 |
| CHEMBL1587502 | — | IC50 | = | 8895.0 | nM | 5.05 |
| CHEMBL1457149 | — | IC50 | = | 12792.0 | nM | 4.89 |
| CHEMBL1700951 | — | IC50 | = | 15008.0 | nM | 4.82 |
| CHEMBL1530437 | — | IC50 | = | 16390.0 | nM | 4.79 |
| CHEMBL1535613 | — | IC50 | = | 19790.0 | nM | 4.70 |
| CHEMBL1399979 | — | IC50 | = | 26629.0 | nM | 4.58 |
| CHEMBL1402286 | — | IC50 | = | 37248.0 | nM | 4.43 |
| CHEMBL1494713 | — | IC50 | > | 50000.0 | nM | - |
| CHEMBL1585333 | — | IC50 | > | 50000.0 | nM | - |
| CHEMBL1399577 | — | IC50 | > | 50000.0 | nM | - |
| CHEMBL1334484 | — | IC50 | > | 50000.0 | nM | - |
| CHEMBL1426689 | — | IC50 | > | 50000.0 | nM | - |
| CHEMBL1507308 | — | IC50 | > | 50000.0 | nM | - |
| CHEMBL1328773 | — | IC50 | > | 50000.0 | nM | - |
| CHEMBL1310699 | — | IC50 | > | 50000.0 | nM | - |
| CHEMBL1481413 | — | IC50 | > | 50000.0 | nM | - |
| CHEMBL1446655 | — | IC50 | > | 50000.0 | nM | - |
| CHEMBL1600114 | — | IC50 | > | 50000.0 | nM | - |
| CHEMBL1404231 | — | IC50 | > | 50000.0 | nM | - |
| CHEMBL1383746 | — | IC50 | > | 50000.0 | nM | - |
| CHEMBL1548870 | — | IC50 | > | 50000.0 | nM | - |