Assay Detail
Functional
CHEMBL1738040
Review assay metadata, readout intent, target linkage, and publication context from the same page.
PUBCHEM_BIOASSAY: Dose Response confirmation of uHTS inhibitors of Mouse Intestinal Alkaline Phosphatase using Placental Alkaline Phosphatase. (Class of assay: confirmatory) [Related pubchem assays (depositor defined):AID2806, AID2818]
134
Total Activities
133
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Category | confirmatory |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Target
Alkaline phosphatase, germ cell type (CHEMBL3402) ↗| Type | SINGLE PROTEIN |
| Organism | Homo sapiens |
Publication
PubChem BioAssay data set
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 134 | 4.64 | 5.63 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL3194421 | — | — | 1 | 5.63 |
| CHEMBL1525897 | — | — | 1 | 5.28 |
| CHEMBL1342091 | — | — | 1 | 5.22 |
| CHEMBL1733511 | — | — | 1 | 5.18 |
| CHEMBL1549540 | — | — | 1 | 5.16 |
| CHEMBL1488474 | — | — | 1 | 5.13 |
| CHEMBL1416189 | — | — | 1 | 5.11 |
| CHEMBL3198600 | — | — | 1 | 5.07 |
| CHEMBL1447139 | — | — | 1 | 4.99 |
| CHEMBL1609295 | — | — | 1 | 4.88 |
| CHEMBL1503852 | — | — | 1 | 4.76 |
| CHEMBL2006611 | — | — | 1 | 4.75 |
| CHEMBL1314122 | — | — | 1 | 4.69 |
| CHEMBL3192085 | — | — | 1 | 4.66 |
| CHEMBL1562260 | — | — | 1 | 4.64 |
| CHEMBL1532097 | DIHYDRODAPHNODORIN B | — | 1 | 4.63 |
| CHEMBL1547446 | — | — | 1 | 4.61 |
| CHEMBL1313502 | — | — | 1 | 4.58 |
| CHEMBL1320230 | — | — | 1 | 4.57 |
| CHEMBL1421399 | — | — | 1 | 4.52 |
| CHEMBL1340344 | — | — | 1 | 4.50 |
| CHEMBL1496952 | — | — | 1 | 4.46 |
| CHEMBL1424867 | — | — | 1 | 4.41 |
| CHEMBL1974737 | — | — | 1 | 4.40 |
| CHEMBL1500102 | — | — | 1 | 4.38 |
| CHEMBL1709713 | — | — | 1 | 4.37 |
| CHEMBL1566994 | — | — | 1 | 4.26 |
| CHEMBL1307435 | — | — | 1 | 4.25 |
| CHEMBL1473059 | — | — | 1 | 4.22 |
| CHEMBL1560432 | — | — | 1 | 4.20 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL3194421 | — | IC50 | = | 2350.0 | nM | 5.63 |
| CHEMBL1525897 | — | IC50 | = | 5310.0 | nM | 5.28 |
| CHEMBL1342091 | — | IC50 | = | 5950.0 | nM | 5.22 |
| CHEMBL1733511 | — | IC50 | = | 6580.0 | nM | 5.18 |
| CHEMBL1549540 | — | IC50 | = | 6940.0 | nM | 5.16 |
| CHEMBL1488474 | — | IC50 | = | 7320.0 | nM | 5.13 |
| CHEMBL1416189 | — | IC50 | = | 7780.0 | nM | 5.11 |
| CHEMBL3198600 | — | IC50 | = | 8440.0 | nM | 5.07 |
| CHEMBL1447139 | — | IC50 | = | 10200.0 | nM | 4.99 |
| CHEMBL1609295 | — | IC50 | = | 13200.0 | nM | 4.88 |
| CHEMBL1503852 | — | IC50 | = | 17200.0 | nM | 4.76 |
| CHEMBL2006611 | — | IC50 | = | 18000.0 | nM | 4.75 |
| CHEMBL1314122 | — | IC50 | = | 20500.0 | nM | 4.69 |
| CHEMBL3192085 | — | IC50 | = | 21800.0 | nM | 4.66 |
| CHEMBL1562260 | — | IC50 | = | 23000.0 | nM | 4.64 |
| CHEMBL1532097 | DIHYDRODAPHNODORIN B | IC50 | = | 23200.0 | nM | 4.63 |
| CHEMBL1547446 | — | IC50 | = | 24400.0 | nM | 4.61 |
| CHEMBL1313502 | — | IC50 | = | 26300.0 | nM | 4.58 |
| CHEMBL1320230 | — | IC50 | = | 27200.0 | nM | 4.57 |
| CHEMBL1421399 | — | IC50 | = | 30500.0 | nM | 4.52 |
| CHEMBL1340344 | — | IC50 | = | 32000.0 | nM | 4.50 |
| CHEMBL1496952 | — | IC50 | = | 34300.0 | nM | 4.46 |
| CHEMBL1424867 | — | IC50 | = | 39400.0 | nM | 4.41 |
| CHEMBL1974737 | — | IC50 | = | 39900.0 | nM | 4.40 |
| CHEMBL1500102 | — | IC50 | = | 42000.0 | nM | 4.38 |
| CHEMBL1709713 | — | IC50 | = | 42500.0 | nM | 4.37 |
| CHEMBL1566994 | — | IC50 | = | 55100.0 | nM | 4.26 |
| CHEMBL1307435 | — | IC50 | = | 56600.0 | nM | 4.25 |
| CHEMBL1473059 | — | IC50 | = | 60200.0 | nM | 4.22 |
| CHEMBL140 | CURCUMIN | IC50 | = | 63500.0 | nM | 4.20 |
| CHEMBL1560432 | — | IC50 | = | 62600.0 | nM | 4.20 |
| CHEMBL1589514 | — | IC50 | = | 64900.0 | nM | 4.19 |
| CHEMBL490355 | SULFURETIN | IC50 | = | 67200.0 | nM | 4.17 |
| CHEMBL1980197 | — | IC50 | = | 70100.0 | nM | 4.15 |
| CHEMBL1375199 | — | IC50 | = | 72700.0 | nM | 4.14 |
| CHEMBL1402586 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL1505816 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL1987928 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL1417524 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL1360321 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL1441918 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL1451040 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL1518080 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL1439675 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL1493010 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL1722786 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL1375627 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL40275 | ALOE-EMODIN | IC50 | > | 100000.0 | nM | - |
| CHEMBL1985299 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL1534899 | — | IC50 | > | 100000.0 | nM | - |