Assay Detail
Functional
CHEMBL1738243
Review assay metadata, readout intent, target linkage, and publication context from the same page.
PUBCHEM_BIOASSAY: Dose Response confirmation of inhibitors of Sentrin-specific proteases (SENPs) using a Luminescent Interference Counterscreen assay. (Class of assay: confirmatory) [Related pubchem assays (depositor defined):AID2540, AID2575, AID2582, AID2599, AID434973, AID434986, AID489001]
27
Total Activities
27
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Category | confirmatory |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
PubChem BioAssay data set
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 27 | 6.11 | 6.49 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL1506796 | — | — | 1 | 6.49 |
| CHEMBL1421255 | — | — | 1 | 6.39 |
| CHEMBL1967857 | — | — | 1 | 6.34 |
| CHEMBL1475128 | — | — | 1 | 6.33 |
| CHEMBL3195102 | — | — | 1 | 6.26 |
| CHEMBL1418096 | — | — | 1 | 6.22 |
| CHEMBL595840 | — | — | 1 | 6.22 |
| CHEMBL1988780 | — | — | 1 | 6.11 |
| CHEMBL1480814 | — | — | 1 | 6.08 |
| CHEMBL1469807 | — | — | 1 | 6.06 |
| CHEMBL1380580 | — | — | 1 | 6.05 |
| CHEMBL281980 | — | — | 1 | 6.05 |
| CHEMBL340701 | — | — | 1 | 5.93 |
| CHEMBL3191962 | — | — | 1 | 5.60 |
| CHEMBL1542328 | — | — | 1 | 5.54 |
| CHEMBL3196451 | — | — | 1 | - |
| CHEMBL1402456 | — | — | 1 | - |
| CHEMBL36536 | — | — | 1 | - |
| CHEMBL1969046 | — | — | 1 | - |
| CHEMBL1471498 | — | — | 1 | - |
| CHEMBL1417815 | — | — | 1 | - |
| CHEMBL205040 | — | — | 1 | - |
| CHEMBL1998302 | — | — | 1 | - |
| CHEMBL1376622 | — | — | 1 | - |
| CHEMBL1449923 | — | — | 1 | - |
| CHEMBL1477061 | — | — | 1 | - |
| CHEMBL1575869 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL1506796 | — | IC50 | = | 325.0 | nM | 6.49 |
| CHEMBL1421255 | — | IC50 | = | 403.0 | nM | 6.39 |
| CHEMBL1967857 | — | IC50 | = | 458.0 | nM | 6.34 |
| CHEMBL1475128 | — | IC50 | = | 471.0 | nM | 6.33 |
| CHEMBL3195102 | — | IC50 | = | 548.0 | nM | 6.26 |
| CHEMBL1418096 | — | IC50 | = | 606.0 | nM | 6.22 |
| CHEMBL595840 | — | IC50 | = | 607.0 | nM | 6.22 |
| CHEMBL1988780 | — | IC50 | = | 782.0 | nM | 6.11 |
| CHEMBL1480814 | — | IC50 | = | 824.0 | nM | 6.08 |
| CHEMBL1469807 | — | IC50 | = | 865.0 | nM | 6.06 |
| CHEMBL1380580 | — | IC50 | = | 888.0 | nM | 6.05 |
| CHEMBL281980 | — | IC50 | = | 884.0 | nM | 6.05 |
| CHEMBL340701 | — | IC50 | = | 1184.0 | nM | 5.93 |
| CHEMBL3191962 | — | IC50 | = | 2532.0 | nM | 5.60 |
| CHEMBL1542328 | — | IC50 | = | 2913.0 | nM | 5.54 |
| CHEMBL3196451 | — | IC50 | > | 5000.0 | nM | - |
| CHEMBL1402456 | — | IC50 | > | 5000.0 | nM | - |
| CHEMBL36536 | — | IC50 | > | 5000.0 | nM | - |
| CHEMBL1969046 | — | IC50 | > | 5000.0 | nM | - |
| CHEMBL1471498 | — | IC50 | > | 5000.0 | nM | - |
| CHEMBL1417815 | — | IC50 | > | 5000.0 | nM | - |
| CHEMBL205040 | — | IC50 | > | 5000.0 | nM | - |
| CHEMBL1998302 | — | IC50 | > | 5000.0 | nM | - |
| CHEMBL1376622 | — | IC50 | > | 5000.0 | nM | - |
| CHEMBL1449923 | — | IC50 | > | 5000.0 | nM | - |
| CHEMBL1477061 | — | IC50 | > | 5000.0 | nM | - |
| CHEMBL1575869 | — | IC50 | > | 5000.0 | nM | - |