Assay Detail
Functional
CHEMBL1738247
Review assay metadata, readout intent, target linkage, and publication context from the same page.
PUBCHEM_BIOASSAY: Dose Response confirmation of uHTS activators of Human Intestinal Alkaline Phosphatase using Mouse Intestinal Alkaline Phosphatase. (Class of assay: confirmatory) [Related pubchem assays (depositor defined):AID2524, AID2571]
44
Total Activities
44
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Mus musculus |
| Category | confirmatory |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Target
Intestinal-type alkaline phosphatase (CHEMBL3151) ↗| Type | SINGLE PROTEIN |
| Organism | Mus musculus |
Publication
PubChem BioAssay data set
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| EC50 | 44 | 4.30 | 4.65 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL1410588 | — | — | 1 | 4.65 |
| CHEMBL1556273 | — | — | 1 | 4.58 |
| CHEMBL1370217 | — | — | 1 | 4.54 |
| CHEMBL1398243 | — | — | 1 | 4.47 |
| CHEMBL1426383 | — | — | 1 | 4.37 |
| CHEMBL1536250 | — | — | 1 | 4.30 |
| CHEMBL1721503 | — | — | 1 | 4.29 |
| CHEMBL1701850 | — | — | 1 | 4.28 |
| CHEMBL1458290 | — | — | 1 | 4.26 |
| CHEMBL1507315 | — | — | 1 | 4.24 |
| CHEMBL1328229 | — | — | 1 | 4.22 |
| CHEMBL1699830 | — | — | 1 | 4.21 |
| CHEMBL1459664 | — | — | 1 | 4.17 |
| CHEMBL1587847 | — | — | 1 | 4.12 |
| CHEMBL1510785 | — | — | 1 | 4.09 |
| CHEMBL1584967 | — | — | 1 | 4.06 |
| CHEMBL1411435 | — | — | 1 | - |
| CHEMBL1348355 | — | — | 1 | - |
| CHEMBL1375639 | — | — | 1 | - |
| CHEMBL3199041 | — | — | 1 | - |
| CHEMBL1528487 | — | — | 1 | - |
| CHEMBL1724929 | — | — | 1 | - |
| CHEMBL1357122 | — | — | 1 | - |
| CHEMBL1463851 | — | — | 1 | - |
| CHEMBL2094652 | — | — | 1 | - |
| CHEMBL1393616 | — | — | 1 | - |
| CHEMBL1707286 | — | — | 1 | - |
| CHEMBL3199008 | — | — | 1 | - |
| CHEMBL1583835 | — | — | 1 | - |
| CHEMBL1352305 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL1410588 | — | EC50 | = | 22400.0 | nM | 4.65 |
| CHEMBL1556273 | — | EC50 | = | 26600.0 | nM | 4.58 |
| CHEMBL1370217 | — | EC50 | = | 28900.0 | nM | 4.54 |
| CHEMBL1398243 | — | EC50 | = | 33900.0 | nM | 4.47 |
| CHEMBL1426383 | — | EC50 | = | 43200.0 | nM | 4.37 |
| CHEMBL1536250 | — | EC50 | = | 49900.0 | nM | 4.30 |
| CHEMBL1721503 | — | EC50 | = | 51300.0 | nM | 4.29 |
| CHEMBL1701850 | — | EC50 | = | 52600.0 | nM | 4.28 |
| CHEMBL1458290 | — | EC50 | = | 55100.0 | nM | 4.26 |
| CHEMBL1507315 | — | EC50 | = | 58200.0 | nM | 4.24 |
| CHEMBL1328229 | — | EC50 | = | 60100.0 | nM | 4.22 |
| CHEMBL1699830 | — | EC50 | = | 61000.0 | nM | 4.21 |
| CHEMBL1459664 | — | EC50 | = | 67500.0 | nM | 4.17 |
| CHEMBL1587847 | — | EC50 | = | 75000.0 | nM | 4.12 |
| CHEMBL1510785 | — | EC50 | = | 80600.0 | nM | 4.09 |
| CHEMBL1584967 | — | EC50 | = | 88000.0 | nM | 4.06 |
| CHEMBL3144972 | — | EC50 | > | 100000.0 | nM | - |
| CHEMBL1386267 | — | EC50 | > | 100000.0 | nM | - |
| CHEMBL1585156 | — | EC50 | > | 100000.0 | nM | - |
| CHEMBL1527436 | — | EC50 | > | 100000.0 | nM | - |
| CHEMBL1719094 | — | EC50 | > | 100000.0 | nM | - |
| CHEMBL1461502 | — | EC50 | > | 100000.0 | nM | - |
| CHEMBL1585596 | — | EC50 | > | 100000.0 | nM | - |
| CHEMBL1399492 | — | EC50 | > | 100000.0 | nM | - |
| CHEMBL195258 | — | EC50 | > | 100000.0 | nM | - |
| CHEMBL3199267 | — | EC50 | > | 100000.0 | nM | - |
| CHEMBL3199528 | — | EC50 | > | 100000.0 | nM | - |
| CHEMBL1721433 | — | EC50 | > | 100000.0 | nM | - |
| CHEMBL1702573 | — | EC50 | > | 100000.0 | nM | - |
| CHEMBL1370019 | — | EC50 | > | 100000.0 | nM | - |
| CHEMBL1352305 | — | EC50 | > | 100000.0 | nM | - |
| CHEMBL1583835 | — | EC50 | > | 100000.0 | nM | - |
| CHEMBL3199008 | — | EC50 | > | 100000.0 | nM | - |
| CHEMBL1707286 | — | EC50 | > | 100000.0 | nM | - |
| CHEMBL1393616 | — | EC50 | > | 100000.0 | nM | - |
| CHEMBL2094652 | — | EC50 | > | 100000.0 | nM | - |
| CHEMBL1463851 | — | EC50 | > | 100000.0 | nM | - |
| CHEMBL1357122 | — | EC50 | > | 100000.0 | nM | - |
| CHEMBL1724929 | — | EC50 | > | 100000.0 | nM | - |
| CHEMBL1528487 | — | EC50 | > | 100000.0 | nM | - |
| CHEMBL3199041 | — | EC50 | > | 100000.0 | nM | - |
| CHEMBL1375639 | — | EC50 | > | 100000.0 | nM | - |
| CHEMBL1348355 | — | EC50 | > | 100000.0 | nM | - |
| CHEMBL1411435 | — | EC50 | > | 100000.0 | nM | - |