Assay Detail
Functional
CHEMBL1738499
Review assay metadata, readout intent, target linkage, and publication context from the same page.
PUBCHEM_BIOASSAY: SAR Confirmatory Dose Response LIBS Assay for Allosteric Ligands of the VLA-4 Integrin. (Class of assay: confirmatory) [Related pubchem assays (depositor defined):AID2557, AID2617, AID2813, AID449766, AID528, AID529]
19
Total Activities
19
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Category | confirmatory |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
PubChem BioAssay data set
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| EC50 | 19 | 5.16 | 6.48 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL163958 | — | — | 1 | 6.48 |
| CHEMBL1361821 | — | — | 1 | 6.47 |
| CHEMBL1388639 | — | — | 1 | 5.62 |
| CHEMBL562729 | — | — | 1 | 5.41 |
| CHEMBL1337800 | — | — | 1 | 5.15 |
| CHEMBL1412583 | — | — | 1 | 4.93 |
| CHEMBL1421490 | — | — | 1 | 4.79 |
| CHEMBL1540682 | — | — | 1 | 4.72 |
| CHEMBL1714669 | — | — | 1 | 4.63 |
| CHEMBL1732679 | — | — | 1 | 4.63 |
| CHEMBL1702298 | — | — | 1 | 4.58 |
| CHEMBL1717333 | — | — | 1 | 4.54 |
| CHEMBL1541441 | — | — | 1 | - |
| CHEMBL1720389 | — | — | 1 | - |
| CHEMBL1521536 | — | — | 1 | - |
| CHEMBL1715259 | — | — | 1 | - |
| CHEMBL1719643 | — | — | 1 | - |
| CHEMBL1735848 | — | — | 1 | - |
| CHEMBL1701004 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL163958 | — | EC50 | = | 334.1 | nM | 6.48 |
| CHEMBL1361821 | — | EC50 | = | 335.2 | nM | 6.47 |
| CHEMBL1388639 | — | EC50 | = | 2425.0 | nM | 5.62 |
| CHEMBL562729 | — | EC50 | = | 3892.0 | nM | 5.41 |
| CHEMBL1337800 | — | EC50 | = | 7143.0 | nM | 5.15 |
| CHEMBL1412583 | — | EC50 | = | 11820.0 | nM | 4.93 |
| CHEMBL1421490 | — | EC50 | = | 16350.0 | nM | 4.79 |
| CHEMBL1540682 | — | EC50 | = | 18860.0 | nM | 4.72 |
| CHEMBL1714669 | — | EC50 | = | 23420.0 | nM | 4.63 |
| CHEMBL1732679 | — | EC50 | = | 23280.0 | nM | 4.63 |
| CHEMBL1702298 | — | EC50 | = | 26140.0 | nM | 4.58 |
| CHEMBL1717333 | — | EC50 | = | 29140.0 | nM | 4.54 |
| CHEMBL1541441 | — | EC50 | > | 49220.0 | nM | - |
| CHEMBL1720389 | — | EC50 | > | 57030.0 | nM | - |
| CHEMBL1521536 | — | EC50 | > | 90770.0 | nM | - |
| CHEMBL1715259 | — | EC50 | > | 49360.0 | nM | - |
| CHEMBL1719643 | — | EC50 | > | 42950.0 | nM | - |
| CHEMBL1735848 | — | EC50 | > | 69840.0 | nM | - |
| CHEMBL1701004 | — | EC50 | > | 30020.0 | nM | - |