Assay Detail
Unclassified
CHEMBL1738515
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PUBCHEM_BIOASSAY: Late stage results from the probe development effort to identify inhibitors of Retinoblastoma Binding Protein 9 (RBBP9): Gel-based Activity-Based Protein Profiling (ABPP) IC50. (Class of assay: confirmatory) [Related pubchem assays (depositor defined):AID1515, AID1537, AID1790, AID2299] Panel member name: Panel member description: RBBP9 IC50 Gel-based ABPP Assay
7
Total Activities
7
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Unclassified |
| Category | confirmatory |
| Confidence | 8 — Homologous single protein target |
| Curated By | Autocuration |
Publication
PubChem BioAssay data set
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 7 | 5.50 | 6.20 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL1092791 | — | — | 1 | 6.20 |
| CHEMBL1093346 | — | — | 1 | 5.72 |
| CHEMBL1092116 | — | — | 1 | 5.30 |
| CHEMBL1092376 | — | — | 1 | 5.24 |
| CHEMBL1092114 | — | — | 1 | 5.04 |
| CHEMBL1092816 | — | — | 1 | - |
| CHEMBL1092115 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL1092791 | — | IC50 | = | 635.0 | nM | 6.20 |
| CHEMBL1093346 | — | IC50 | = | 1900.0 | nM | 5.72 |
| CHEMBL1092116 | — | IC50 | = | 5000.0 | nM | 5.30 |
| CHEMBL1092376 | — | IC50 | = | 5700.0 | nM | 5.24 |
| CHEMBL1092114 | — | IC50 | = | 9100.0 | nM | 5.04 |
| CHEMBL1092816 | — | IC50 | = | 1500000.0 | nM | - |
| CHEMBL1092115 | — | IC50 | = | 1200000.0 | nM | - |