Assay Detail
Functional
CHEMBL1738599
Review assay metadata, readout intent, target linkage, and publication context from the same page.
PUBCHEM_BIOASSAY: Dose response counterscreen of uHTS chemical inhibitors of both B-cell and T-cell specific antigen receptor-induced NF-kB activation in a HEK-293T cell line using a luminescence assay. (Class of assay: confirmatory) [Related pubchem assays (depositor defined):AID435003, AID435022, AID465, AID489019, AID489029]
168
Total Activities
168
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Cell Type | HEK-293T |
| Category | confirmatory |
| Confidence | 0 — Uncurated / Unknown |
| Curated By | Autocuration |
Publication
PubChem BioAssay data set
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 168 | 5.74 | 6.77 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL1513566 | — | — | 1 | 6.77 |
| CHEMBL1537098 | — | — | 1 | 6.77 |
| CHEMBL1370991 | — | — | 1 | 6.75 |
| CHEMBL1511219 | — | — | 1 | 6.70 |
| CHEMBL1607801 | — | — | 1 | 6.70 |
| CHEMBL1394722 | — | — | 1 | 6.68 |
| CHEMBL1372292 | — | — | 1 | 6.68 |
| CHEMBL1430094 | — | — | 1 | 6.66 |
| CHEMBL1340715 | — | — | 1 | 6.66 |
| CHEMBL1422572 | — | — | 1 | 6.62 |
| CHEMBL1524484 | — | — | 1 | 6.62 |
| CHEMBL513000 | — | — | 1 | 6.58 |
| CHEMBL1425552 | — | — | 1 | 6.58 |
| CHEMBL1440954 | — | — | 1 | 6.57 |
| CHEMBL1584044 | — | — | 1 | 6.55 |
| CHEMBL1728497 | — | — | 1 | 6.51 |
| CHEMBL1441604 | — | — | 1 | 6.51 |
| CHEMBL1575502 | — | — | 1 | 6.50 |
| CHEMBL1569724 | — | — | 1 | 6.50 |
| CHEMBL1430096 | — | — | 1 | 6.48 |
| CHEMBL1567944 | — | — | 1 | 6.48 |
| CHEMBL1329446 | — | — | 1 | 6.42 |
| CHEMBL300389 | — | — | 1 | 6.42 |
| CHEMBL1729737 | — | — | 1 | 6.42 |
| CHEMBL1513705 | — | — | 1 | 6.42 |
| CHEMBL3189250 | — | — | 1 | 6.39 |
| CHEMBL1499501 | — | — | 1 | 6.36 |
| CHEMBL1521023 | — | — | 1 | 6.36 |
| CHEMBL1358722 | — | — | 1 | 6.35 |
| CHEMBL1360997 | — | — | 1 | 6.34 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL1513566 | — | IC50 | = | 170.0 | nM | 6.77 |
| CHEMBL1537098 | — | IC50 | = | 170.0 | nM | 6.77 |
| CHEMBL1370991 | — | IC50 | = | 180.0 | nM | 6.75 |
| CHEMBL1607801 | — | IC50 | = | 200.0 | nM | 6.70 |
| CHEMBL1511219 | — | IC50 | = | 200.0 | nM | 6.70 |
| CHEMBL1394722 | — | IC50 | = | 210.0 | nM | 6.68 |
| CHEMBL1372292 | — | IC50 | = | 210.0 | nM | 6.68 |
| CHEMBL1430094 | — | IC50 | = | 220.0 | nM | 6.66 |
| CHEMBL1340715 | — | IC50 | = | 220.0 | nM | 6.66 |
| CHEMBL1422572 | — | IC50 | = | 240.0 | nM | 6.62 |
| CHEMBL1524484 | — | IC50 | = | 240.0 | nM | 6.62 |
| CHEMBL513000 | — | IC50 | = | 260.0 | nM | 6.58 |
| CHEMBL1425552 | — | IC50 | = | 260.0 | nM | 6.58 |
| CHEMBL1440954 | — | IC50 | = | 270.0 | nM | 6.57 |
| CHEMBL1584044 | — | IC50 | = | 280.0 | nM | 6.55 |
| CHEMBL1441604 | — | IC50 | = | 310.0 | nM | 6.51 |
| CHEMBL1728497 | — | IC50 | = | 310.0 | nM | 6.51 |
| CHEMBL1569724 | — | IC50 | = | 320.0 | nM | 6.50 |
| CHEMBL1575502 | — | IC50 | = | 320.0 | nM | 6.50 |
| CHEMBL1430096 | — | IC50 | = | 330.0 | nM | 6.48 |
| CHEMBL1567944 | — | IC50 | = | 330.0 | nM | 6.48 |
| CHEMBL1329446 | — | IC50 | = | 380.0 | nM | 6.42 |
| CHEMBL1729737 | — | IC50 | = | 380.0 | nM | 6.42 |
| CHEMBL1513705 | — | IC50 | = | 380.0 | nM | 6.42 |
| CHEMBL300389 | — | IC50 | = | 380.0 | nM | 6.42 |
| CHEMBL3189250 | — | IC50 | = | 410.0 | nM | 6.39 |
| CHEMBL1499501 | — | IC50 | = | 440.0 | nM | 6.36 |
| CHEMBL1521023 | — | IC50 | = | 440.0 | nM | 6.36 |
| CHEMBL1358722 | — | IC50 | = | 450.0 | nM | 6.35 |
| CHEMBL1360997 | — | IC50 | = | 460.0 | nM | 6.34 |
| CHEMBL1491705 | — | IC50 | = | 470.0 | nM | 6.33 |
| CHEMBL1304342 | — | IC50 | = | 470.0 | nM | 6.33 |
| CHEMBL1432721 | — | IC50 | = | 470.0 | nM | 6.33 |
| CHEMBL601933 | — | IC50 | = | 510.0 | nM | 6.29 |
| CHEMBL1310617 | — | IC50 | = | 550.0 | nM | 6.26 |
| CHEMBL1544743 | — | IC50 | = | 560.0 | nM | 6.25 |
| CHEMBL1308223 | — | IC50 | = | 600.0 | nM | 6.22 |
| CHEMBL1302130 | — | IC50 | = | 600.0 | nM | 6.22 |
| CHEMBL1712104 | — | IC50 | = | 610.0 | nM | 6.21 |
| CHEMBL1490293 | — | IC50 | = | 610.0 | nM | 6.21 |
| CHEMBL1386804 | — | IC50 | = | 610.0 | nM | 6.21 |
| CHEMBL1382917 | — | IC50 | = | 630.0 | nM | 6.20 |
| CHEMBL1404493 | — | IC50 | = | 640.0 | nM | 6.19 |
| CHEMBL1382191 | — | IC50 | = | 770.0 | nM | 6.11 |
| CHEMBL1459468 | — | IC50 | = | 800.0 | nM | 6.10 |
| CHEMBL1543215 | — | IC50 | = | 790.0 | nM | 6.10 |
| CHEMBL1519965 | — | IC50 | = | 870.0 | nM | 6.06 |
| CHEMBL1549500 | — | IC50 | = | 880.0 | nM | 6.06 |
| CHEMBL1378232 | — | IC50 | = | 900.0 | nM | 6.05 |
| CHEMBL81782 | — | IC50 | = | 940.0 | nM | 6.03 |