Assay Detail
Binding
CHEMBL1763073
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Inhibition of human ERG
13
Total Activities
13
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Target
Voltage-gated inwardly rectifying potassium channel KCNH2 (CHEMBL240) ↗| Type | SINGLE PROTEIN |
| Organism | Homo sapiens |
Publication
The discovery of novel, potent and highly selective inhibitors of inducible nitric oxide synthase (iNOS).
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 13 | 6.00 | 7.00 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL447183 | — | — | 1 | 7.00 |
| CHEMBL1762472 | — | — | 1 | 5.00 |
| CHEMBL1762470 | — | — | 1 | - |
| CHEMBL1762471 | — | — | 1 | - |
| CHEMBL1762473 | — | — | 1 | - |
| CHEMBL1762474 | — | — | 1 | - |
| CHEMBL1762475 | — | — | 1 | - |
| CHEMBL1762476 | — | — | 1 | - |
| CHEMBL1762477 | — | — | 1 | - |
| CHEMBL1762478 | — | — | 1 | - |
| CHEMBL1762479 | — | — | 1 | - |
| CHEMBL1762480 | — | — | 1 | - |
| CHEMBL1762481 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL447183 | — | IC50 | = | 100.0 | nM | 7.00 |
| CHEMBL1762472 | — | IC50 | = | 10000.0 | nM | 5.00 |
| CHEMBL1762470 | — | IC50 | - | — | - | |
| CHEMBL1762471 | — | IC50 | - | — | - | |
| CHEMBL1762473 | — | IC50 | - | — | - | |
| CHEMBL1762474 | — | IC50 | - | — | - | |
| CHEMBL1762475 | — | IC50 | - | — | - | |
| CHEMBL1762476 | — | IC50 | - | — | - | |
| CHEMBL1762477 | — | IC50 | - | — | - | |
| CHEMBL1762478 | — | IC50 | - | — | - | |
| CHEMBL1762479 | — | IC50 | > | 10000.0 | nM | - |
| CHEMBL1762480 | — | IC50 | - | — | - | |
| CHEMBL1762481 | — | IC50 | > | 10000.0 | nM | - |