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Assay Detail

CHEMBL1775502

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Functional
Antiviral activity against Hepatitis C virus infected in human Ava5 cells expressing EG(delta4AB)SEAP reporter gene assessed as decreased viral replication measured as SEAP activity by Phospha-Light assay
2
Total Activities
1
Compounds Tested
2
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Organism Hepacivirus hominis
Cell Type Ava5
Confidence 1 — Organism
Curated By Autocuration

Target

Hepatitis C virus (CHEMBL379)
Type ORGANISM
Organism Hepacivirus hominis

Publication

Diosgenin, a plant-derived sapogenin, exhibits antiviral activity in vitro against hepatitis C virus.
Wang YJ, Pan KL, Hsieh TC, Chang TY, Lin WH, Hsu JT.
J Nat Prod (2011) 74 : 580 -584
PubMed 21391660 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
Activity 1 - -
EC50 1 5.42 5.42

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL412437 DISOGENIN 2 5.42

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL412437 DISOGENIN EC50 = 3800.0 nM 5.42
CHEMBL412437 DISOGENIN Activity - -