Assay Detail
Functional
CHEMBL1794348
Review assay metadata, readout intent, target linkage, and publication context from the same page.
PUBCHEM_BIOASSAY: Dose response counterscreen of uHTS hits for ATG4B inhibitors in a Phospholipase A2 assay Set 2. (Class of assay: confirmatory) [Related pubchem assays (depositor defined):AID504462, AID504475]
16
Total Activities
16
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Category | confirmatory |
| Confidence | 8 — Homologous single protein target |
| Curated By | Autocuration |
Publication
PubChem BioAssay data set
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 16 | 4.67 | 5.61 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL1986418 | — | — | 1 | 5.61 |
| CHEMBL3195142 | — | — | 1 | 5.26 |
| CHEMBL1974450 | — | — | 1 | 4.98 |
| CHEMBL1520424 | — | — | 1 | 4.97 |
| CHEMBL1349405 | — | — | 1 | 4.96 |
| CHEMBL1365132 | — | — | 1 | 4.87 |
| CHEMBL1393538 | — | — | 1 | 4.75 |
| CHEMBL3196472 | — | — | 1 | 4.65 |
| CHEMBL1424479 | — | — | 1 | 4.46 |
| CHEMBL602126 | — | — | 1 | 4.40 |
| CHEMBL1351421 | — | — | 1 | 4.33 |
| CHEMBL1584985 | — | — | 1 | 4.31 |
| CHEMBL1340058 | — | — | 1 | 4.29 |
| CHEMBL1541554 | — | — | 1 | 4.13 |
| CHEMBL1540150 | — | — | 1 | 4.10 |
| CHEMBL1388951 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL1986418 | — | IC50 | = | 2470.0 | nM | 5.61 |
| CHEMBL3195142 | — | IC50 | = | 5500.0 | nM | 5.26 |
| CHEMBL1974450 | — | IC50 | = | 10500.0 | nM | 4.98 |
| CHEMBL1520424 | — | IC50 | = | 10700.0 | nM | 4.97 |
| CHEMBL1349405 | — | IC50 | = | 11100.0 | nM | 4.96 |
| CHEMBL1365132 | — | IC50 | = | 13400.0 | nM | 4.87 |
| CHEMBL1393538 | — | IC50 | = | 17700.0 | nM | 4.75 |
| CHEMBL3196472 | — | IC50 | = | 22300.0 | nM | 4.65 |
| CHEMBL1424479 | — | IC50 | = | 35100.0 | nM | 4.46 |
| CHEMBL602126 | — | IC50 | = | 40100.0 | nM | 4.40 |
| CHEMBL1351421 | — | IC50 | = | 46400.0 | nM | 4.33 |
| CHEMBL1584985 | — | IC50 | = | 48900.0 | nM | 4.31 |
| CHEMBL1340058 | — | IC50 | = | 51700.0 | nM | 4.29 |
| CHEMBL1541554 | — | IC50 | = | 74100.0 | nM | 4.13 |
| CHEMBL1540150 | — | IC50 | = | 79100.0 | nM | 4.10 |
| CHEMBL1388951 | — | IC50 | > | 80000.0 | nM | - |