Assay Detail
Functional
CHEMBL1794477
Review assay metadata, readout intent, target linkage, and publication context from the same page.
PUBCHEM_BIOASSAY: SAR analysis of small molecule inhibitors of hexokinase domain containing I (HKDC1) in the hexokinase 1 selectivity assay. (Class of assay: confirmatory) [Related pubchem assays (depositor defined):AID493160, AID493190]
90
Total Activities
89
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Category | confirmatory |
| Confidence | 8 — Homologous single protein target |
| Curated By | Autocuration |
Publication
PubChem BioAssay data set
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 90 | 4.40 | 5.42 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL1347253 | — | — | 1 | 5.42 |
| CHEMBL1888104 | — | — | 1 | 4.39 |
| CHEMBL1417992 | — | — | 1 | 4.30 |
| CHEMBL1868007 | — | — | 1 | 4.30 |
| CHEMBL1877532 | — | — | 1 | 4.22 |
| CHEMBL1872978 | — | — | 1 | 4.21 |
| CHEMBL1898878 | — | — | 1 | 4.18 |
| CHEMBL1875709 | — | — | 1 | 4.16 |
| CHEMBL1898021 | — | — | 1 | - |
| CHEMBL1903920 | — | — | 1 | - |
| CHEMBL1877088 | — | — | 1 | - |
| CHEMBL1899387 | — | — | 1 | - |
| CHEMBL1895627 | — | — | 1 | - |
| CHEMBL1875828 | — | — | 1 | - |
| CHEMBL1363086 | — | — | 1 | - |
| CHEMBL1505625 | — | — | 1 | - |
| CHEMBL1880882 | — | — | 1 | - |
| CHEMBL1883114 | — | — | 1 | - |
| CHEMBL1903921 | — | — | 1 | - |
| CHEMBL1558854 | — | — | 1 | - |
| CHEMBL1877469 | — | — | 1 | - |
| CHEMBL1877571 | — | — | 1 | - |
| CHEMBL1901046 | — | — | 1 | - |
| CHEMBL1901426 | — | — | 1 | - |
| CHEMBL1900041 | — | — | 1 | - |
| CHEMBL1465938 | — | — | 1 | - |
| CHEMBL1879611 | — | — | 1 | - |
| CHEMBL1900318 | — | — | 1 | - |
| CHEMBL1895705 | — | — | 1 | - |
| CHEMBL1879859 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL1347253 | — | IC50 | = | 3760.0 | nM | 5.42 |
| CHEMBL1888104 | — | IC50 | = | 40300.0 | nM | 4.39 |
| CHEMBL1417992 | — | IC50 | = | 50300.0 | nM | 4.30 |
| CHEMBL1868007 | — | IC50 | = | 50600.0 | nM | 4.30 |
| CHEMBL1877532 | — | IC50 | = | 59800.0 | nM | 4.22 |
| CHEMBL1872978 | — | IC50 | = | 62400.0 | nM | 4.21 |
| CHEMBL1898878 | — | IC50 | = | 65300.0 | nM | 4.18 |
| CHEMBL1875709 | — | IC50 | = | 69000.0 | nM | 4.16 |
| CHEMBL1901940 | — | IC50 | > | 80000.0 | nM | - |
| CHEMBL1903920 | — | IC50 | > | 80000.0 | nM | - |
| CHEMBL1880038 | — | IC50 | > | 80000.0 | nM | - |
| CHEMBL1880647 | — | IC50 | > | 80000.0 | nM | - |
| CHEMBL1905037 | — | IC50 | > | 80000.0 | nM | - |
| CHEMBL1492662 | — | IC50 | > | 80000.0 | nM | - |
| CHEMBL1904466 | — | IC50 | > | 80000.0 | nM | - |
| CHEMBL1884740 | — | IC50 | > | 80000.0 | nM | - |
| CHEMBL1883547 | — | IC50 | > | 80000.0 | nM | - |
| CHEMBL1904169 | — | IC50 | > | 80000.0 | nM | - |
| CHEMBL1889188 | — | IC50 | > | 80000.0 | nM | - |
| CHEMBL1902190 | — | IC50 | > | 80000.0 | nM | - |
| CHEMBL1418314 | — | IC50 | > | 80000.0 | nM | - |
| CHEMBL1882018 | — | IC50 | > | 80000.0 | nM | - |
| CHEMBL1881953 | — | IC50 | > | 80000.0 | nM | - |
| CHEMBL1903268 | — | IC50 | > | 80000.0 | nM | - |
| CHEMBL1903537 | — | IC50 | > | 80000.0 | nM | - |
| CHEMBL1882595 | — | IC50 | > | 80000.0 | nM | - |
| CHEMBL1880360 | — | IC50 | > | 80000.0 | nM | - |
| CHEMBL1334787 | — | IC50 | > | 80000.0 | nM | - |
| CHEMBL1887735 | — | IC50 | > | 80000.0 | nM | - |
| CHEMBL1558854 | — | IC50 | > | 80000.0 | nM | - |
| CHEMBL1879859 | — | IC50 | > | 80000.0 | nM | - |
| CHEMBL1895705 | — | IC50 | > | 80000.0 | nM | - |
| CHEMBL1900318 | — | IC50 | > | 80000.0 | nM | - |
| CHEMBL1879611 | — | IC50 | > | 80000.0 | nM | - |
| CHEMBL1465938 | — | IC50 | > | 80000.0 | nM | - |
| CHEMBL1900041 | — | IC50 | > | 80000.0 | nM | - |
| CHEMBL1901426 | — | IC50 | > | 80000.0 | nM | - |
| CHEMBL1901046 | — | IC50 | > | 80000.0 | nM | - |
| CHEMBL1877571 | — | IC50 | > | 80000.0 | nM | - |
| CHEMBL1877469 | — | IC50 | > | 80000.0 | nM | - |
| CHEMBL1903921 | — | IC50 | > | 80000.0 | nM | - |
| CHEMBL1898021 | — | IC50 | > | 80000.0 | nM | - |
| CHEMBL1877088 | — | IC50 | > | 80000.0 | nM | - |
| CHEMBL1899387 | — | IC50 | > | 80000.0 | nM | - |
| CHEMBL1895627 | — | IC50 | > | 80000.0 | nM | - |
| CHEMBL1875828 | — | IC50 | > | 80000.0 | nM | - |
| CHEMBL1363086 | — | IC50 | > | 80000.0 | nM | - |
| CHEMBL1896660 | — | IC50 | > | 80000.0 | nM | - |
| CHEMBL1880882 | — | IC50 | > | 80000.0 | nM | - |
| CHEMBL1883114 | — | IC50 | > | 80000.0 | nM | - |