Skip to main content
Free research Free research Free assay review with research home and workspace preview
Quick search ChEMBL 36
Assay Detail

CHEMBL1804265

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Binding
Binding affinity to chimpanzee P2Y14 receptor
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Binding
Organism Pan troglodytes
Confidence 0 — Uncurated / Unknown
Curated By Autocuration

Target

Unchecked (CHEMBL612545)
Type UNCHECKED

Publication

Applying the pro-drug approach to afford highly bioavailable antagonists of P2Y(14).
Robichaud J, Fournier JF, Gagné S, Gauthier JY, Hamel M, Han Y, Hénault M, Kargman S, Levesque JF, Mamane Y, Mancini J, Morin N, Mulrooney E, Wu J, Black WC.
Bioorg Med Chem Lett (2011) 21 : 4366 -4368
PubMed 21689930 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
Ki 2 8.56 8.72

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL1800685 PPTN 1 8.72
CHEMBL1774903 1 8.40

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL1800685 PPTN Ki = 1.9 nM 8.72
CHEMBL1774903 Ki = 4.0 nM 8.40