Assay Detail
Functional
CHEMBL1805405
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Agonist activity at GPR109a
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Confidence | 8 — Homologous single protein target |
| Curated By | Autocuration |
Publication
Progress in structure based drug design for G protein-coupled receptors.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| EC50 | 2 | 5.66 | 6.42 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL1802361 | — | — | 1 | 6.42 |
| CHEMBL228244 | — | — | 1 | 4.90 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL1802361 | — | EC50 | = | 380.0 | nM | 6.42 |
| CHEMBL228244 | — | EC50 | = | 12500.0 | nM | 4.90 |