Assay Detail
Binding
CHEMBL1814965
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Inhibition of PARP-1 using [32P]-NAD+ after 15 mins
9
Total Activities
9
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Confidence | 8 — Homologous single protein target |
| Curated By | Autocuration |
Publication
Discovery and structure-activity relationships of modified salicylanilides as cell permeable inhibitors of poly(ADP-ribose) glycohydrolase (PARG).
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 9 | 4.56 | 5.27 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL267373 | BENZAMIDE | — | 1 | 5.27 |
| CHEMBL115114 | — | — | 1 | 4.66 |
| CHEMBL1813887 | — | — | 1 | 4.18 |
| CHEMBL1813880 | — | — | 1 | 4.11 |
| CHEMBL1813879 | — | — | 1 | - |
| CHEMBL1813881 | — | — | 1 | - |
| CHEMBL1814050 | — | — | 1 | - |
| CHEMBL1814051 | — | — | 1 | - |
| CHEMBL1230692 | ADENOSINE DIPHOSPHATE (HYDROXYMETHYL)PYRROLIDINEDIOL | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL267373 | BENZAMIDE | IC50 | = | 5400.0 | nM | 5.27 |
| CHEMBL115114 | — | IC50 | = | 22000.0 | nM | 4.66 |
| CHEMBL1813887 | — | IC50 | = | 66000.0 | nM | 4.18 |
| CHEMBL1813880 | — | IC50 | = | 78000.0 | nM | 4.11 |
| CHEMBL1813879 | — | IC50 | = | 123000.0 | nM | - |
| CHEMBL1813881 | — | IC50 | = | 120000.0 | nM | - |
| CHEMBL1814050 | — | IC50 | = | 500000.0 | nM | - |
| CHEMBL1814051 | — | IC50 | = | 500000.0 | nM | - |
| CHEMBL1230692 | ADENOSINE DIPHOSPHATE (HYDROXYMETHYL)PYRROLIDINEDIOL | IC50 | > | 1000000.0 | nM | - |