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Assay Detail

CHEMBL1817164

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Functional
Antiviral activity against HCV JFH-1 assessed as inhibition of viral replication by cell based assay
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Organism Hepacivirus hominis
Confidence 1 — Organism
Curated By Autocuration

Target

Hepatitis C virus (CHEMBL379)
Type ORGANISM
Organism Hepacivirus hominis

Publication

Discovery of naturally occurring aurones that are potent allosteric inhibitors of hepatitis C virus RNA-dependent RNA polymerase.
Haudecoeur R, Ahmed-Belkacem A, Yi W, Fortuné A, Brillet R, Belle C, Nicolle E, Pallier C, Pawlotsky JM, Boumendjel A.
J Med Chem (2011) 54 : 5395 -5402
PubMed 21699179 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 2 4.58 4.75

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL199975 1 4.75
CHEMBL201626 1 4.40

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL199975 IC50 = 18000.0 nM 4.75
CHEMBL201626 IC50 = 40000.0 nM 4.40