Assay Detail
Binding
CHEMBL1820097
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Inhibition of JNK1 expressed in Escherichia coli or baculovirus-infected insect cells by TR-FRET assay
4
Total Activities
3
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Confidence | 8 — Homologous single protein target |
| Curated By | Autocuration |
Publication
Selectivity of kinase inhibitor fragments.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 4 | 7.55 | 7.55 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL243298 | — | — | 1 | 7.55 |
| CHEMBL389685 | — | — | 2 | - |
| CHEMBL1817872 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL243298 | — | IC50 | = | 28.0 | nM | 7.55 |
| CHEMBL389685 | — | IC50 | > | 667000.0 | nM | - |
| CHEMBL1817872 | — | IC50 | < | 500.0 | nM | - |
| CHEMBL389685 | — | IC50 | > | 630957.34 | nM | - |