Assay Detail
Functional
CHEMBL1825337
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Agonist activity at human TRPv1 receptor expressed in HEK293 cells assessed as stimulation of intracellular calcium level using Fluo4-AM dye based fluorimetric assay
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Cell Type | HEK293 |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Target
Transient receptor potential cation channel subfamily V member 1 (CHEMBL4794) ↗| Type | SINGLE PROTEIN |
| Organism | Homo sapiens |
Publication
Bioactive prenylogous cannabinoid from fiber hemp (Cannabis sativa).
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| EC50 | 2 | 5.63 | 5.89 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL497318 | CANNABIGEROL | 2.0 | 1 | 5.89 |
| CHEMBL1823117 | SESQUICANNABIGEROL | — | 1 | 5.36 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL497318 | CANNABIGEROL | EC50 | = | 1300.0 | nM | 5.89 |
| CHEMBL1823117 | SESQUICANNABIGEROL | EC50 | = | 4400.0 | nM | 5.36 |