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Assay Detail

CHEMBL1825489

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Functional
Antiproliferative activity against human A549 cells assessed as loss of cell viability after 48 hrs by MTT assay
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Organism Homo sapiens
Cell Type A549
Confidence 1 — Organism
Curated By Autocuration

Target

A549 (CHEMBL392)
Type CELL-LINE
Organism Homo sapiens

Publication

Curcumin recognizes a unique binding site of tubulin.
Chakraborti S, Das L, Kapoor N, Das A, Dwivedi V, Poddar A, Chakraborti G, Janik M, Basu G, Panda D, Chakrabarti P, Surolia A, Bhattacharyya B.
J Med Chem (2011) 54 : 6183 -6196
PubMed 21830815 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 2 4.97 5.16

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL428441 1 5.16
CHEMBL140 CURCUMIN 3.0 1 4.77

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL428441 IC50 = 7000.0 nM 5.16
CHEMBL140 CURCUMIN IC50 = 17000.0 nM 4.77