Assay Detail
Functional
CHEMBL1827052
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Antifungal activity against Candida albicans isolate CaCi-2 after 48 hrs by Almar blue fluorimetry
16
Total Activities
16
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Candida albicans |
| Confidence | 1 — Organism |
| Curated By | Autocuration |
Publication
Piperazinyl quinolines as chemosensitizers to increase fluconazole susceptibility of Candida albicans clinical isolates.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 16 | 4.82 | 4.82 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL1360505 | — | — | 1 | 4.82 |
| CHEMBL1256729 | — | — | 1 | 4.82 |
| CHEMBL1822266 | — | — | 1 | 4.82 |
| CHEMBL1822267 | — | — | 1 | 4.82 |
| CHEMBL1822268 | — | — | 1 | 4.82 |
| CHEMBL1822269 | — | — | 1 | 4.82 |
| CHEMBL1822270 | — | — | 1 | 4.82 |
| CHEMBL1822271 | — | — | 1 | 4.82 |
| CHEMBL1822272 | — | — | 1 | 4.82 |
| CHEMBL1822273 | — | — | 1 | 4.82 |
| CHEMBL1822274 | — | — | 1 | 4.82 |
| CHEMBL1585578 | — | — | 1 | 4.82 |
| CHEMBL1822275 | — | — | 1 | 4.82 |
| CHEMBL1822276 | — | — | 1 | 4.82 |
| CHEMBL1822277 | — | — | 1 | 4.82 |
| CHEMBL1822278 | — | — | 1 | 4.82 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL1360505 | — | IC50 | = | 15000.0 | nM | 4.82 |
| CHEMBL1256729 | — | IC50 | = | 15000.0 | nM | 4.82 |
| CHEMBL1822266 | — | IC50 | = | 15000.0 | nM | 4.82 |
| CHEMBL1822267 | — | IC50 | = | 15000.0 | nM | 4.82 |
| CHEMBL1822268 | — | IC50 | = | 15000.0 | nM | 4.82 |
| CHEMBL1822269 | — | IC50 | = | 15000.0 | nM | 4.82 |
| CHEMBL1822270 | — | IC50 | = | 15000.0 | nM | 4.82 |
| CHEMBL1822271 | — | IC50 | = | 15000.0 | nM | 4.82 |
| CHEMBL1822272 | — | IC50 | = | 15000.0 | nM | 4.82 |
| CHEMBL1822273 | — | IC50 | = | 15000.0 | nM | 4.82 |
| CHEMBL1822274 | — | IC50 | = | 15000.0 | nM | 4.82 |
| CHEMBL1585578 | — | IC50 | = | 15000.0 | nM | 4.82 |
| CHEMBL1822275 | — | IC50 | = | 15000.0 | nM | 4.82 |
| CHEMBL1822276 | — | IC50 | = | 15000.0 | nM | 4.82 |
| CHEMBL1822277 | — | IC50 | = | 15000.0 | nM | 4.82 |
| CHEMBL1822278 | — | IC50 | = | 15000.0 | nM | 4.82 |