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Assay Detail

CHEMBL1827928

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Binding
Inhibition of quorum sensing Salmonella Typhimurium by beta-galactosidase transcription assay in presence of 50 uM DPD
6
Total Activities
6
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Binding
Organism Salmonella enterica subsp. enterica serovar Typhimurium
Confidence 0 — Uncurated / Unknown
Curated By Autocuration

Target

Unchecked (CHEMBL612545)
Type UNCHECKED

Publication

Medicinal chemistry as a conduit for the modulation of quorum sensing.
Lowery CA, Salzameda NT, Sawada D, Kaufmann GF, Janda KD.
J Med Chem (2010) 53 : 7467 -7489
PubMed 20669927 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 6 4.97 5.30

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL539143 1 5.30
CHEMBL539221 1 5.28
CHEMBL1824157 1 4.69
CHEMBL550518 1 4.60
CHEMBL1824156 1 -
CHEMBL560745 1 -

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL539143 IC50 = 5040.0 nM 5.30
CHEMBL539221 IC50 = 5300.0 nM 5.28
CHEMBL1824157 IC50 = 20300.0 nM 4.69
CHEMBL550518 IC50 = 24900.0 nM 4.60
CHEMBL1824156 IC50 > 50000.0 nM -
CHEMBL560745 IC50 > 50000.0 nM -