Assay Detail
Binding
CHEMBL1839748
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Inhibition of human recombinant MMP7 assessed as hydrolysis of MOCAcPLGLA2pr(Dnp)AR-NH2 by fluorescence spectrofluorometry
3
Total Activities
3
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
Selective water-soluble gelatinase inhibitor prodrugs.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ki | 3 | 4.41 | 4.41 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL485492 | — | — | 1 | 4.41 |
| CHEMBL1834420 | — | — | 1 | - |
| CHEMBL1834423 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL485492 | — | Ki | = | 39000.0 | nM | 4.41 |
| CHEMBL1834420 | — | Ki | = | 160000.0 | nM | - |
| CHEMBL1834423 | — | Ki | = | 116000.0 | nM | - |