Assay Detail
Functional
CHEMBL1912153
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Antibiofilm activity against Paracoccus sp. 4M6 assessed as inhibition of bacterial adhesion after 15 hrs by fluorescence assay
22
Total Activities
22
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Paracoccus sp. |
| Confidence | 1 — Organism |
| Curated By | Autocuration |
Publication
Designing 2-aminoimidazole alkaloids analogs with anti-biofilm activities: structure-activities relationships of polysubstituted triazoles.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| EC50 | 22 | 4.21 | 4.38 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL1910932 | — | — | 1 | 4.38 |
| CHEMBL1910926 | — | — | 1 | 4.04 |
| CHEMBL1910823 | — | — | 1 | - |
| CHEMBL1910824 | — | — | 1 | - |
| CHEMBL1910825 | — | — | 1 | - |
| CHEMBL1910826 | — | — | 1 | - |
| CHEMBL1910827 | — | — | 1 | - |
| CHEMBL1910923 | — | — | 1 | - |
| CHEMBL1910924 | — | — | 1 | - |
| CHEMBL1910925 | — | — | 1 | - |
| CHEMBL1514247 | — | — | 1 | - |
| CHEMBL1910822 | — | — | 1 | - |
| CHEMBL1910928 | — | — | 1 | - |
| CHEMBL1910921 | — | — | 1 | - |
| CHEMBL1910922 | — | — | 1 | - |
| CHEMBL1910929 | — | — | 1 | - |
| CHEMBL1910930 | — | — | 1 | - |
| CHEMBL1910931 | — | — | 1 | - |
| CHEMBL1910933 | — | — | 1 | - |
| CHEMBL1910934 | — | — | 1 | - |
| CHEMBL1910935 | — | — | 1 | - |
| CHEMBL1910927 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL1910932 | — | EC50 | = | 41200.0 | nM | 4.38 |
| CHEMBL1910926 | — | EC50 | = | 90300.0 | nM | 4.04 |
| CHEMBL1910823 | — | EC50 | > | 200000.0 | nM | - |
| CHEMBL1910824 | — | EC50 | > | 200000.0 | nM | - |
| CHEMBL1910825 | — | EC50 | = | 199300.0 | nM | - |
| CHEMBL1910826 | — | EC50 | > | 200000.0 | nM | - |
| CHEMBL1910827 | — | EC50 | > | 200000.0 | nM | - |
| CHEMBL1910923 | — | EC50 | > | 200000.0 | nM | - |
| CHEMBL1910924 | — | EC50 | > | 200000.0 | nM | - |
| CHEMBL1910925 | — | EC50 | > | 200000.0 | nM | - |
| CHEMBL1514247 | — | EC50 | > | 200000.0 | nM | - |
| CHEMBL1910822 | — | EC50 | > | 200000.0 | nM | - |
| CHEMBL1910928 | — | EC50 | > | 200000.0 | nM | - |
| CHEMBL1910921 | — | EC50 | = | 199300.0 | nM | - |
| CHEMBL1910922 | — | EC50 | > | 200000.0 | nM | - |
| CHEMBL1910929 | — | EC50 | > | 200000.0 | nM | - |
| CHEMBL1910930 | — | EC50 | > | 200000.0 | nM | - |
| CHEMBL1910931 | — | EC50 | > | 200000.0 | nM | - |
| CHEMBL1910933 | — | EC50 | > | 200000.0 | nM | - |
| CHEMBL1910934 | — | EC50 | = | 130800.0 | nM | - |
| CHEMBL1910935 | — | EC50 | = | 181100.0 | nM | - |
| CHEMBL1910927 | — | EC50 | > | 200000.0 | nM | - |