Assay Detail
Binding
CHEMBL1936809
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Inhibition of dopamine D2 receptor
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Confidence | 8 — Homologous single protein target |
| Curated By | Autocuration |
Publication
Discovery and characterization of a potent and selective antagonist of melanin-concentrating hormone receptor 2.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 2 | 6.06 | 6.30 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL1934127 | — | — | 1 | 6.30 |
| CHEMBL1934130 | — | — | 1 | 5.82 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL1934127 | — | IC50 | = | 500.0 | nM | 6.30 |
| CHEMBL1934130 | — | IC50 | = | 1500.0 | nM | 5.82 |