Assay Detail
Binding
CHEMBL1942541
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Inhibition of PHD1
3
Total Activities
3
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Confidence | 8 — Homologous single protein target |
| Curated By | Autocuration |
Publication
Lysine demethylases inhibitors.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 3 | 4.98 | 5.68 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL90852 | N-OXALYLGLYCINE | — | 1 | 5.68 |
| CHEMBL1938900 | — | — | 1 | 4.27 |
| CHEMBL1229308 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL90852 | N-OXALYLGLYCINE | IC50 | = | 2100.0 | nM | 5.68 |
| CHEMBL1938900 | — | IC50 | = | 54000.0 | nM | 4.27 |
| CHEMBL1229308 | — | IC50 | > | 100000.0 | nM | - |