Assay Detail
Binding
CHEMBL1947809
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Binding affinity to Alpha-1D adrenoceptor expressed in HEK cells by calcium flux assay
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Cell Type | HEK293 |
| Confidence | 8 — Homologous single protein target |
| Curated By | Autocuration |
Publication
From libraries to candidate: the discovery of new ultra long-acting dibasic β₂-adrenoceptor agonists.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| EC50 | 1 | 6.90 | 6.90 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL1945039 | — | — | 1 | 6.90 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL1945039 | — | EC50 | = | 125.89 | nM | 6.90 |