Assay Detail
Binding
CHEMBL1961271
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Competitive inhibition of human CSNK2A1/2B by Lineweaver-Burk plot analysis in presence of cosubstrate ATP
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 7 — Homologous single protein target |
| Curated By | Autocuration |
Publication
Indeno[1,2-b]indole derivatives as a novel class of potent human protein kinase CK2 inhibitors.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ki | 1 | 6.82 | 6.82 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL1957190 | — | — | 1 | 6.82 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL1957190 | — | Ki | = | 150.0 | nM | 6.82 |