Assay Detail
Functional
CHEMBL1963962
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PUBCHEM_BIOASSAY: SAR analysis of small molecule inhibitors of Apaf-1 using a LZ-Caspase-9/Caspase-3 Fluorescent Selectivity assay. (Class of assay: confirmatory)
22
Total Activities
22
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Category | confirmatory |
| Confidence | 0 — Uncurated / Unknown |
| Curated By | Autocuration |
Publication
PubChem BioAssay data set
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 22 | 4.14 | 4.43 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL1985990 | — | — | 1 | 4.43 |
| CHEMBL1098875 | — | — | 1 | 4.39 |
| CHEMBL2369351 | — | — | 1 | 4.14 |
| CHEMBL2006389 | — | — | 1 | 4.07 |
| CHEMBL1969075 | — | — | 1 | 4.05 |
| CHEMBL307480 | — | — | 1 | 4.05 |
| CHEMBL1538897 | — | — | 1 | 4.01 |
| CHEMBL1979370 | — | — | 1 | 4.00 |
| CHEMBL1969207 | — | — | 1 | - |
| CHEMBL2369347 | — | — | 1 | - |
| CHEMBL1343853 | — | — | 1 | - |
| CHEMBL1427763 | — | — | 1 | - |
| CHEMBL1525481 | — | — | 1 | - |
| CHEMBL1540627 | — | — | 1 | - |
| CHEMBL600336 | — | — | 1 | - |
| CHEMBL312537 | — | — | 1 | - |
| CHEMBL1310325 | — | — | 1 | - |
| CHEMBL1981019 | — | — | 1 | - |
| CHEMBL1382209 | — | — | 1 | - |
| CHEMBL2004532 | — | — | 1 | - |
| CHEMBL2005851 | — | — | 1 | - |
| CHEMBL1978889 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL1985990 | — | IC50 | = | 37500.0 | nM | 4.43 |
| CHEMBL1098875 | — | IC50 | = | 40900.0 | nM | 4.39 |
| CHEMBL2369351 | — | IC50 | = | 72000.0 | nM | 4.14 |
| CHEMBL2006389 | — | IC50 | = | 85300.0 | nM | 4.07 |
| CHEMBL1969075 | — | IC50 | = | 89700.0 | nM | 4.05 |
| CHEMBL307480 | — | IC50 | = | 89600.0 | nM | 4.05 |
| CHEMBL1538897 | — | IC50 | = | 97300.0 | nM | 4.01 |
| CHEMBL1979370 | — | IC50 | = | 98800.0 | nM | 4.00 |
| CHEMBL1969207 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL2369347 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL1343853 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL1427763 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL1525481 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL1540627 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL600336 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL312537 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL1310325 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL1981019 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL1382209 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL2004532 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL2005851 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL1978889 | — | IC50 | > | 100000.0 | nM | - |